SCHEMBL17525014

SCHEMBL17525014

Cc1cc(Nc2ccc(N3CCC4(CC3)C(=O)Nc3ncccc34)nc2)cc(C)n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CALCA P06881 4/20 0.38
CRBN Q96SW2 1/20 0.37
CALCRL Q16602 7/20 0.35
ADM2 Q7Z4H4 4/20 0.35
CALCB P10092 3/20 0.35
KCNH2 Q12809 1/20 0.35
CACNA1C Q13936 1/20 0.35
ASIC3 Q9UHC3 1/20 0.35
JAK1 P23458 3/20 0.34
JAK3 P52333 3/20 0.34
JAK2 O60674 2/20 0.34
TYK2 P29597 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524984 0.91 CALCRL (0.35) CALCACALCRLADM2CALCB
SCHEMBL17525112 0.83 SCN9A (0.43) CALCACRBNCALCRL
SCHEMBL17524992 0.82 CALCA (0.39) CALCACRBNKCNH2
SCHEMBL17524906 0.81 CALCA (0.40) CALCACALCRLKCNH2
SCHEMBL17506417 0.78 CALCA (0.40) CALCACRBNCALCRLKCNH2CYP3A4
SCHEMBL17524937 0.78 ME2 (0.40) CALCACRBNCALCRLKCNH2
SCHEMBL17525060 0.75 MAPT (0.39) JAK1JAK3JAK2TYK2
SCHEMBL17524879 0.75 HTR6 (0.34) CALCA
SCHEMBL17524997 0.74 EGLN1 (0.43) CALCACALCRLKCNH2
SCHEMBL17524875 0.74 NPC1 (0.45) CALCACALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed