SCHEMBL17524910

SCHEMBL17524910

Cc1ccc(N2CCC3(CC2)C(=O)Nc2ncccc23)cc1C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 4/20 0.43
ADRB1 P08588 1/20 0.42
CALCA P06881 4/20 0.41
KDM4E B2RXH2 1/20 0.40
DRD4 P21917 7/20 0.39
DRD2 P14416 6/20 0.39
DRD3 P35462 4/20 0.39
HTR1A P08908 2/20 0.37
HTR2A P28223 2/20 0.37
HTR7 P34969 2/20 0.37
HTR6 P50406 1/20 0.37
ADRA2C P18825 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17525077 0.91 HTR7 (0.46) CALCAHTR1AHTR2AHTR7HTR6
SCHEMBL17524935 0.91 GAA (0.44) EGLN1CALCAHTR1AHTR2AHTR7
SCHEMBL17524994 0.90 CALCRL (0.40) EGLN1CALCAHTR1AHTR2AHTR7
SCHEMBL17524907 0.88 MALT1 (0.41) EGLN1CALCAKDM4ELMNA
SCHEMBL17524901 0.86 ADRA2B (0.40) EGLN1CALCAHTR1AHTR2AHTR7
SCHEMBL17524997 0.85 EGLN1 (0.43) EGLN1CALCADRD3HTR1AHTR2A
SCHEMBL17525019 0.84 MAPK1 (0.41) CALCADRD4HTR1AHTR2AHTR7
SCHEMBL17524923 0.83 CALCA (0.41) CALCAKDM4EHTR1AHTR2AHTR7
SCHEMBL17525079 0.83 KCNH2 (0.38) EGLN1CALCAHTR1AHTR2AHTR7
SCHEMBL17524909 0.83 ADRA1A (0.38) EGLN1CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed