SCHEMBL17524935

SCHEMBL17524935

Cc1cc(N2CCC3(CC2)C(=O)Nc2ncccc23)ccc1N

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.44
RAD52 P43351 1/20 0.44
CALCA P06881 4/20 0.40
EGLN1 Q9GZT9 8/20 0.37
HTR7 P34969 3/20 0.36
HTR1A P08908 2/20 0.36
HTR2A P28223 2/20 0.36
HTR6 P50406 2/20 0.36
CALCB P10092 1/20 0.35
ADM2 Q7Z4H4 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
CALCRL Q16602 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524910 0.91 EGLN1 (0.43) CALCAEGLN1HTR7HTR1AHTR2A
SCHEMBL17525077 0.87 HTR7 (0.46) CALCAHTR7HTR1AHTR2AHTR6
SCHEMBL17524938 0.87 HTR7 (0.45) CALCAHTR7HTR1AHTR2AHTR6
SCHEMBL17524940 0.87 CALCA (0.40) CALCAHTR7HTR1AHTR2AHTR6
SCHEMBL17524933 0.86 CALCA (0.40) CALCAEGLN1HTR7HTR1AHTR2A
SCHEMBL17524994 0.86 CALCRL (0.40) CALCAEGLN1HTR7HTR1AHTR2A
SCHEMBL17524942 0.84 ADRA2B (0.40) CALCAEGLN1HTR7HTR1AHTR2A
SCHEMBL17524907 0.84 MALT1 (0.41) CALCAEGLN1MALT1CALCRL
SCHEMBL17524923 0.83 CALCA (0.41) GAARAD52CALCAHTR7HTR1A
SCHEMBL17524997 0.83 EGLN1 (0.43) CALCAEGLN1HTR7HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed