SCHEMBL17524907

SCHEMBL17524907

COc1cc(N2CCC3(CC2)C(=O)Nc2ncccc23)ccc1C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 1/20 0.41
MAP3K11 Q16584 1/20 0.39
CALCA P06881 3/20 0.38
EGLN1 Q9GZT9 3/20 0.38
TGFBR1 P36897 1/20 0.38
ACVR1 Q04771 1/20 0.38
PDE4B Q07343 1/20 0.37
CALCRL Q16602 2/20 0.37
TNK2 Q07912 3/20 0.37
AVPR1A P37288 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
IDH1 O75874 1/20 0.35
DPP4 P27487 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524901 0.90 ADRA2B (0.40) MALT1CALCAEGLN1CALCRLALDH1A1
SCHEMBL17524933 0.90 CALCA (0.40) MALT1MAP3K11CALCAEGLN1CALCRL
SCHEMBL17524910 0.88 EGLN1 (0.43) CALCAEGLN1LMNAKDM4E
SCHEMBL17525080 0.86 LRRK2 (0.39) CALCAEGLN1CALCRL
SCHEMBL17525079 0.86 KCNH2 (0.38) CALCAEGLN1CALCRLIDH1
SCHEMBL17524909 0.86 ADRA1A (0.38) CALCAEGLN1CALCRLIDH1
SCHEMBL17525077 0.86 HTR7 (0.46) MALT1CALCAALDH1A1LMNA
SCHEMBL17524994 0.85 CALCRL (0.40) CALCAEGLN1PDE4BCALCRL
SCHEMBL17524935 0.84 GAA (0.44) MALT1CALCAEGLN1CALCRL
SCHEMBL17524942 0.82 ADRA2B (0.40) CALCAEGLN1CALCRLTNK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed