SCHEMBL17524879

SCHEMBL17524879

Cc1cc(Nc2ccc(N3CCC4(CC3)C(=O)Nc3ncccc34)cc2Oc2ccccc2)cc(C)n1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.34
TNK2 Q07912 11/20 0.34
CALCA P06881 2/20 0.34
MAPK7 Q13164 1/20 0.34
LRRK2 Q5S007 1/20 0.34
MAPK10 P53779 1/20 0.33
IGF1R P08069 3/20 0.33
EGLN1 Q9GZT9 1/20 0.33
EGFR P00533 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524873 0.82 HTR6 (0.38) HTR6CALCAEGLN1
SCHEMBL17524928 0.81 HTR6 (0.37) HTR6CALCAEGLN1
SCHEMBL17524881 0.79 CRHR1 (0.33) HTR6CALCAEGLN1
SCHEMBL17524907 0.75 MALT1 (0.41) TNK2CALCAEGLN1
SCHEMBL17525014 0.75 CALCA (0.38) CALCA
SCHEMBL17524875 0.75 NPC1 (0.45) CALCA
SCHEMBL17525080 0.74 LRRK2 (0.39) HTR6CALCALRRK2EGLN1
SCHEMBL17524901 0.74 ADRA2B (0.40) HTR6CALCAEGLN1
SCHEMBL17524910 0.74 EGLN1 (0.43) HTR6CALCAEGLN1
SCHEMBL17524933 0.73 CALCA (0.40) HTR6CALCAEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed