SCHEMBL1754860

SCHEMBL1754860

CC(N(c1ccc2nccnc2c1)S(=O)(=O)c1cc(Cl)cc(Cl)c1)P(=O)(O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD11B1 P28845 2/20 0.34
ATM Q13315 1/20 0.34
NPC1 O15118 4/20 0.31
RAB9A P51151 4/20 0.31
KMT2A Q03164 2/20 0.31
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31
HTT P42858 1/20 0.30
S1PR1 P21453 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
PSEN1 P49768 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1754893 0.88 MMP2 (0.41) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL2055490 0.79 S1PR1 (0.38) ATMNPC1RAB9AKMT2AHTT
SCHEMBL3277899 0.78 KDR (0.40) ALDH1A1KDM4EHPGDHSD17B10NPC1
SCHEMBL1754859 0.77 S1PR1 (0.37) HPGDATMNPC1RAB9AKMT2A
SCHEMBL1754852 0.76 NR3C1 (0.41) MAPTNPC1KMT2AMEN1
SCHEMBL2098568 0.75 ATM (0.32) ATMNPC1RAB9AS1PR1
SCHEMBL3803818 0.73 AHR (0.42) MAPTKMT2AMEN1
SCHEMBL2055376 0.73 S1PR1 (0.35) ALDH1A1KDM4EMAPTATMRAB9A
SCHEMBL3278252 0.73 SLC40A1 (0.40) ALDH1A1KDM4ETP53MAPTKMT2A
SCHEMBL3277708 0.68 ACLY (0.32) HSD11B1MMP2MMP13PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200987-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2010-06-30 EP claimed
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO claimed
EP-2200987-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2010-06-30 EP disclosed
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO disclosed