SCHEMBL3277899

SCHEMBL3277899

CC(N(c1cnc2ccccc2c1)S(=O)(=O)c1cc(Cl)cc(Cl)c1)P(=O)(O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
ALPL P05186 6/20 0.40
MMP2 P08253 1/20 0.39
MMP13 P45452 1/20 0.39
TMPRSS4 Q9NRS4 1/20 0.39
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
TRPM8 Q7Z2W7 1/20 0.36
HTR6 P50406 2/20 0.36
HTR2C P28335 1/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BCAT1 P54687 1/20 0.35
MET P08581 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1754893 0.86 MMP2 (0.41) KDRMMP2MMP13ALDH1A1HTR6
SCHEMBL2055486 0.80 S1PR1 (0.42) KDRCNR1CNR2ALPLMMP2
SCHEMBL3277898 0.78 S1PR1 (0.40) KDRCNR1CNR2ALPLMMP2
SCHEMBL1754860 0.78 ALDH1A1 (0.35) MMP2MMP13KDM4EALDH1A1NPC1
SCHEMBL3278252 0.77 SLC40A1 (0.40) KDRCNR1KDM4EALDH1A1TSHR
SCHEMBL3277708 0.77 ACLY (0.32) MMP2MMP13HTR6
SCHEMBL1754852 0.77 NR3C1 (0.41) HTR6NPC1L3MBTL1
SCHEMBL2101977 0.76 CNR2 (0.40) KDRCNR1CNR2ALPLMMP2
SCHEMBL2055378 0.74 RAB9A (0.41) KDRCNR1CNR2ALPLKDM4E
SCHEMBL3281740 0.72 PSEN1 (0.35) MMP2HTR6HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200987-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2010-06-30 EP disclosed
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO disclosed