SCHEMBL3277708

SCHEMBL3277708

CC(N(c1cccc2cncnc12)S(=O)(=O)c1cc(Cl)cc(Cl)c1)P(=O)(O)O

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.32
HTR6 P50406 1/20 0.32
ITGA4 P13612 1/20 0.32
GRM4 Q14833 1/20 0.32
HSD11B1 P28845 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
ABCB1 P08183 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP3 P08254 1/20 0.30
MMP7 P09237 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30
MMP13 P45452 1/20 0.30
MMP14 P50281 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3278252 0.87 SLC40A1 (0.40) ABCB1
SCHEMBL1754210 0.82 MEN1 (0.35) ACLYGRM4
SCHEMBL1754854 0.80 MEN1 (0.33) ACLYHSD11B1PSEN1PSEN2APH1B
SCHEMBL3277703 0.80 MEN1 (0.35) ACLYITGA4
SCHEMBL3277899 0.77 KDR (0.40) HTR6MMP2MMP13
SCHEMBL2055406 0.76 MEN1 (0.33)
SCHEMBL1754852 0.76 NR3C1 (0.41) ACLYHTR6
SCHEMBL3281740 0.73 PSEN1 (0.35) ACLYHTR6HSD11B1PSEN1PSEN2
SCHEMBL1754893 0.72 MMP2 (0.41) HTR6MMP2MMP13
SCHEMBL1754867 0.72 ALDH1A1 (0.37) ACLYHSD11B1PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200987-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2010-06-30 EP disclosed
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO disclosed