SCHEMBL17563243

SCHEMBL17563243

CN1C(=O)OCc2ccc(S(C)(=O)=O)cc21

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PNMT P11086 3/20 0.38
PTGS2 P35354 9/20 0.35
PTGS1 P23219 6/20 0.35
ALDH1A1 P00352 2/20 0.35
ABCB11 O95342 1/20 0.35
MT-CO2 P00403 1/20 0.35
HTR1A P08908 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
MC4R P32245 1/20 0.35
KDM1A O60341 1/20 0.35
GAA P10253 1/20 0.34
TRIM24 O15164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15833697 0.87 ALDH1A1 (0.33) ALDH1A1GAATRIM24
SCHEMBL13091165 0.78 HSD17B10 (0.40) ALDH1A1GAA
SCHEMBL31714457 0.76 LMNA (0.45) ALDH1A1GAA
SCHEMBL12698059 0.76 POLB (0.41)
SCHEMBL31714699 0.75 CASP1 (0.49) ALDH1A1GAA
SCHEMBL10075473 0.74 PKM (0.61) ALDH1A1GAATRIM24
SCHEMBL10076590 0.73 DRD2 (0.52) ALDH1A1GAATRIM24
SCHEMBL5423529 0.72 MAOA (0.44)
SCHEMBL30525088 0.71 ALDH1A1 (0.51) PTGS2PTGS1ALDH1A1ABCB11MT-CO2
SCHEMBL20791320 0.71 ALDH1A1 (0.51) PTGS2PTGS1ALDH1A1ABCB11MT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655350-B1 BICYCLIC PKM2 ACTIVATORS AGIOS PHARMACEUTICALS INC (US) 2016-03-09 EP disclosed