SCHEMBL1758

SCHEMBL1758

CCCC(=O)C1(c2ccc(Cl)cc2)CCC1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.51
HSD11B1 P28845 8/20 0.51
NCOA1 Q15788 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
GAA P10253 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
OPRM1 P35372 1/20 0.45
ALDH1A1 P00352 4/20 0.44
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
THRB P10828 1/20 0.43
MAPK1 P28482 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2421 0.91 HSD11B1 (0.49) HDAC4HSD11B1NCOA1SMN1; SMN2CHRM2
SCHEMBL2550 0.87 HDAC4 (0.54) HDAC4HSD11B1NCOA1SMN1; SMN2CHRM2
SCHEMBL12980674 0.84 ALDH1A1 (0.43) HDAC4HSD11B1OPRM1ALDH1A1MEN1
SCHEMBL2023 0.83 OPRM1 (0.48) CHRM2CHRM1OPRM1
SCHEMBL13267655 0.82 HDAC4 (0.57) HDAC4HSD11B1SMN1; SMN2CHRM2CHRM1
SCHEMBL3443916 0.81 HDAC4 (0.56) HDAC4HSD11B1NCOA1SMN1; SMN2ALDH1A1
SCHEMBL1770373 0.81 HDAC4 (0.56) HDAC4HSD11B1NCOA1SMN1; SMN2ALDH1A1
SCHEMBL8225678 0.80 HDAC4 (0.54) HDAC4HSD11B1NCOA1SMN1; SMN2ALDH1A1
SCHEMBL1769960 0.80 HDAC4 (0.54) HDAC4HSD11B1SMN1; SMN2CHRM2CHRM1
SCHEMBL13545175 0.80 HSD11B1 (0.51) HDAC4HSD11B1SMN1; SMN2CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4814352-A ANTIDEPRESSANT CYCLOBUTYL BENZYLAMINE THE BOOTS COMPANY PLC (GB) 1989-03-21 US disclosed
US-4806570-A ANTIDEPRESSANTS THE BOOTS COMPANY PLC (GB) 1989-02-21 US disclosed
US-4767790-A ANTIDEPRESSANTS THE BOOTS COMPANY PLC (GB) 1988-08-30 US disclosed
US-4746680-A ANTIDEPRESSANTS THE BOOTS COMPANY P.L.C. (GB) 1988-05-24 US disclosed
US-4522828-A CYCLOBUTYLALKYLAMINE COMPOUNDS, ANTIDEPRESSANTS THE BOOTS COMPANY PLC (GB) 1985-06-11 US disclosed