SCHEMBL17595142

SCHEMBL17595142

CCc1cc(C(=O)OC(=O)c2c(O)c(CC)c(-c3ccc(N4CCN(C(=O)OC(C)(C)C)CC4)cc3)[nH]c2=O)c(=O)[nH]c1-c1ccc(N2CCNCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.39
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
ALK Q9UM73 1/20 0.35
TLR9 Q9NR96 2/20 0.35
TLR8 Q9NR97 2/20 0.35
TLR7 Q9NYK1 2/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP2C19 P33261 1/20 0.34
EZH2 Q15910 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NAMPT P43490 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17595141 0.90 ABCB1 (0.40) ABCB1DDB1CRBNLMNAMAPT
SCHEMBL17594871 0.85 ALDH1A1 (0.39) LMNAMAPTALDH1A1TLR9TLR8
SCHEMBL17594971 0.84 LMNA (0.39) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL14746007 0.82 MAPT (0.45) ABCB1DDB1CRBNLMNAMAPT
SCHEMBL17595032 0.82 LMNA (0.42) DDB1CRBNLMNAMAPTALDH1A1
SCHEMBL14745432 0.80 MAPT (0.47) DDB1CRBNLMNAMAPTALDH1A1
SCHEMBL14744882 0.75 EZH2 (0.38) MAPTTLR9TLR8TLR7EZH2
SCHEMBL14758613 0.75 TLR9 (0.42) ABCB1ALDH1A1TLR9TLR8TLR7
SCHEMBL17595028 0.74 ALDH1A1 (0.42) DDB1CRBNLMNAMAPTALDH1A1
SCHEMBL17595256 0.74 PDE3B (0.35) LMNAMAPTALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed