SCHEMBL1765201

SCHEMBL1765201

NCc1cc(F)cc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.46
LOXL2 Q9Y4K0 3/20 0.42
IDO1 P14902 4/20 0.38
DAO P14920 2/20 0.37
TAAR1 Q96RJ0 4/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36
MAOB P27338 2/20 0.35
S100A9 P06702 1/20 0.35
METAP2 P50579 1/20 0.35
LOX P28300 1/20 0.34
LOXL3 P58215 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237616 0.82 TAAR1 (0.50) PNMTTAAR1MAOB
SCHEMBL111874 0.82 PNMT (0.56) PNMTLOXL2IDO1TAAR1CSNK2B
SCHEMBL43006 0.82 LOXL2 (0.52) LOXL2IDO1TAAR1MAOB
SCHEMBL625883 0.82 PNMT (0.56) PNMTLOXL2IDO1TAAR1CSNK2B
Hydrochloric Acid SCHEMBL12521203 0.80 TAAR1 (0.48) PNMTIDO1TAAR1MAOB
Hydrochloric Acid SCHEMBL2457582 0.79 IDO1 (0.54) LOXL2IDO1TAAR1MAOB
SCHEMBL14750162 0.78 DAO (0.38) IDO1DAOS100A9METAP2
SCHEMBL31322887 0.78 DAO (0.38) IDO1DAOS100A9METAP2
SCHEMBL857310 0.76 DAO (0.37) IDO1DAOS100A9METAP2
SCHEMBL146087 0.76 DAO (0.37) IDO1DAOS100A9METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627631-B1 PYRROLIDINONES AS METAP2 INHIBITORS MERCK PATENT GMBH (DE) 2015-12-16 EP claimed
US-8895535-B2 Pyrrolidinones as MetAP-2 inhibitors MERCK PATENT GMBH (DE) 2014-11-25 US claimed
US-20130296274-A1 PYRROLIDINONES AS METAP-2 INHIBITORS MERCK PATENT GMBH (DE) 2013-11-07 US claimed
EP-4612131-A1 NICOTINAMIDE DERIVATIVES FOR USE IN TREATING DISORDERS ASSOCIATED WITH KCNK13 ACTIVITY Cerevance, Inc. (US) 2025-09-10 EP disclosed
CN-116768824-B Imide azole heterocyclic compound and application thereof 华南农业大学 2025-06-10 CN disclosed
WO-2024119838-A1 IMIDAZOLE HETEROCYCLIC COMPOUND AND USE THEREOF 华南农业大学 2024-06-13 WO disclosed
WO-2024095003-A1 NICOTINAMIDE DERIVATIVES FOR USE IN TREATING DISORDERS ASSOCIATED WITH KCNK13 ACTIVITY Cerevance, Inc. (US) 2024-05-10 WO disclosed
EP-3609868-B1 TETRAHYDROQUINOLINE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS RAQUALIA PHARMA INC (JP) 2023-10-18 EP disclosed
EP-3307727-B1 HETEROCYCLIC INHIBITORS OF ERK1 AND ERK2 AND THEIR USE IN THE TREATMENT OF CANCER ASANA BIOSCIENCES LLC (US) 2023-10-04 EP disclosed
CN-116768824-A Imide azole heterocyclic compound and application thereof 华南农业大学 2023-09-19 CN disclosed
WO-2023154291-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed
WO-2012048775-A1 PYRROLIDINONES AS METAP2 INHIBITORS MERCK PATENT GMBH (DE) 2012-04-19 WO disclosed
WO-2011064141-A1 SULTAM DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-06-03 WO disclosed
US-20110124686-A1 SULTAM DERIVATIVES ANDERSON KEVIN W 2011-05-26 US disclosed
US-7442692-B2 Indanyl-piperazine compounds LES LABORATOIRES SERVIER (FR) 2008-10-28 US disclosed
WO-2006103342-A9 INDANYL-PIPERAZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2007-10-25 WO disclosed
EP-1707564-B1 Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2007-09-12 EP disclosed
US-20060223830-A1 Indanyl-piperazine compounds LES LABORATOIRES SERVIER (FR) 2006-10-05 US disclosed
WO-2006103342-A2 INDANYL-PIPERAZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2006-10-05 WO disclosed
EP-1707564-A2 Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2006-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060223830-A1 Indanyl-piperazine compounds HTR4, NR4A1, NR4A3 PNMT 551/4885LOXL2 3963/4885IDO1 315/4885
US-20130296274-A1 PYRROLIDINONES AS METAP-2 INHIBITORS METAP1, METAP2, DNPEP PNMT 139/4885LOXL2 1739/4885IDO1 187/4885
US-20110124686-A1 SULTAM DERIVATIVES SULT1A1, SULT2A1, SULT1E1 PNMT 355/4885LOXL2 4252/4885IDO1 575/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.