SCHEMBL17656375

SCHEMBL17656375

N#CCc1ccc2c(c1)CCC(F)(F)CC2

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.37
ESR1 P03372 6/20 0.37
ENPP2 Q13822 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
MMP3 P08254 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4521078 0.82 ENPP2 (0.39) ENPP2MMP3KDM4ETDP1
SCHEMBL1466419 0.80 RXRB (0.40) ENPP2MMP3KDM4ETDP1
SCHEMBL16526955 0.77 ESR1 (0.31) ESR2ESR1
SCHEMBL17656382 0.75 KDM1A (0.34) ESR2ESR1ENPP2
SCHEMBL21218921 0.72 ENPP2 (0.40) ESR2ESR1ENPP2L3MBTL1MMP3
SCHEMBL28840767 0.70 PRMT5 (0.38) ENPP2MMP3KDM4ETDP1
SCHEMBL17656383 0.70 OPRM1 (0.40)
SCHEMBL1789393 0.69 NPC1 (0.40) ESR2ESR1L3MBTL1KDM4E
SCHEMBL29790934 0.68 ENPP2 (0.37) ENPP2L3MBTL1MMP3KDM4ETDP1
SCHEMBL27582186 0.68 ENPP2 (0.37) ENPP2L3MBTL1MMP3KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2674428-B1 Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2016-04-06 EP disclosed