Maleic Acid

Maleic Acid

SCHEMBL1766045

C=CC(=O)OCC.C=COC(C)=O.O=C(O)/C=C\C(=O)O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.56
TSHR P16473 7/20 0.41
HPGD P15428 1/20 0.41
ALDH1A1 P00352 6/20 0.38
HSD17B10 Q99714 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 3/20 0.36
HIF1A Q16665 3/20 0.36
CYP3A4 P08684 2/20 0.36
THRB P10828 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acrylic Acid Ethyl Ester SCHEMBL11043394 0.93 HCAR2 (0.46) HCAR2TSHRHPGDALDH1A1HSD17B10
Ethyl Fumarate SCHEMBL9678685 0.92 HCAR2 (0.69) HCAR2ALDH1A1HSD17B10LMNANPSR1
Ethyl Fumarate SCHEMBL9678697 0.92 HCAR2 (0.69) HCAR2ALDH1A1HSD17B10LMNANPSR1
Acrylic Acid Ethyl Ester SCHEMBL8060405 0.91 TSHR (0.47) HCAR2TSHRHPGDALDH1A1HSD17B10
Ethyl Fumarate SCHEMBL10900161 0.89 HCAR2 (0.65) HCAR2ALDH1A1HSD17B10LMNANPSR1
Acrylic Acid Ethyl Ester SCHEMBL28542637 0.88 TSHR (0.44) HCAR2TSHRHPGDALDH1A1HSD17B10
Maleic Acid SCHEMBL5400251 0.88 HCAR2 (0.58) HCAR2TSHRHPGDALDH1A1LMNA
Fumaric Acid SCHEMBL8925070 0.88 HCAR2 (0.72) HCAR2TSHRHPGDALDH1A1HSD17B10
Fumaric Acid SCHEMBL10717454 0.88 HCAR2 (0.72) HCAR2TSHRHPGDALDH1A1HSD17B10
Maleic Acid SCHEMBL8772268 0.88 HCAR2 (0.72) HCAR2TSHRHPGDALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106103359-A Compositions and methods for fouling control in regulated vaporization systems 索理思科技开曼公司 2016-11-09 CN claimed
US-8530403-B2 Solidification matrix using a maleic-containing terpolymer binding agent ECOLAB USA INC. (US) 2013-09-10 US claimed
US-10737221-B2 Scale inhibitor for reverse osmosis membranes and reverse osmosis membrane treatment method KURITA WATER INDUSTRIES LTD. (JP) 2020-08-11 US disclosed
US-20190030489-A1 SCALE INHIBITOR FOR REVERSE OSMOSIS MEMBRANES AND REVERSE OSMOSIS MEMBRANE TREATMENT METHOD KURITA WATER INDUSTRIES LTD. (JP) 2019-01-31 US disclosed
US-20160046515-A1 METHOD FOR PREVENTING SCALE DEPOSITION AND SCALE INHIBITOR KURITA WATER INDUSTRIES LTD. (JP) 2016-02-18 US disclosed
US-8530403-B2 Solidification matrix using a maleic-containing terpolymer binding agent ECOLAB USA INC. (US) 2013-09-10 US disclosed
US-20110124546-A1 SOLIDIFICATION MATRIX USING A MALEIC-CONTAINING TERPOLYMER BINDING AGENT ECOLAB INC. (US) 2011-05-26 US disclosed
WO-2011061654-A2 SOLIDIFICATION MATRIX USING A MALEIC-CONTAINING TERPOLYMER BINDING AGENT ECOLAB INC. (US) 2011-05-26 WO disclosed