SCHEMBL17664358

SCHEMBL17664358

Fc1ccc(Cc2ccc(Cl)cn2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PARP1 P09874 2/20 0.40
IDO1 P14902 1/20 0.40
HTR1A P08908 3/20 0.39
GRM4 Q14833 1/20 0.36
PIK3CA P42336 1/20 0.36
HSP90AB1 P08238 1/20 0.36
EGFR P00533 2/20 0.36
GPR52 Q9Y2T5 1/20 0.35
CYP3A4 P08684 1/20 0.35
SLC6A4 P31645 2/20 0.35
HTR2A P28223 1/20 0.35
KCNH2 Q12809 1/20 0.35
SOS1 Q07889 1/20 0.35
DAO P14920 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17664001 0.89 GPR52 (0.35) HDAC3HDAC1HDAC2HDAC6PARP1
SCHEMBL17664100 0.88 FYN (0.41) HSP90AB1DAO
SCHEMBL17663857 0.86 IDO1 (0.42) IDO1HSP90AB1CYP3A4SLC6A4
SCHEMBL23716265 0.84 RXRA (0.39) HSP90AB1SLC6A4HTR2AKCNH2DAO
SCHEMBL23716215 0.83 MBOAT4 (0.37) HSP90AB1CYP3A4SLC6A4HTR2AKCNH2
SCHEMBL23716203 0.82 MBOAT4 (0.39) HSP90AB1CYP3A4SLC6A4HTR2AKCNH2
SCHEMBL17663971 0.80 HSP90AB1 (0.47) IDO1HSP90AB1
SCHEMBL29442805 0.77 ALDH1A1 (0.54) HDAC3HDAC1HDAC2HDAC6PARP1
SCHEMBL21384002 0.77 ALDH1A1 (0.54) HDAC3HDAC1HDAC2HDAC6PARP1
SCHEMBL17664376 0.76 ALDH1A1 (0.43) IDO1HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed
WO-2016053855-A1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-04-07 WO disclosed