SCHEMBL1768148

SCHEMBL1768148

CC1COC2(CCNCC2)O1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2489261 1.00 HTR1A (0.34) HTR1AADRA1DADRA1AADRA1B
SCHEMBL9739360 0.88
SCHEMBL3308565 0.79 PABPC1 (0.42) HTR1AADRA1DADRA1AADRA1B
SCHEMBL14272690 0.79
SCHEMBL10265045 0.79
SCHEMBL12662822 0.79
SCHEMBL3305308 0.77 PABPC1 (0.44) HTR1AADRA1DADRA1AADRA1B
SCHEMBL12944468 0.77 PABPC1 (0.44) HTR1AADRA1DADRA1AADRA1B
SCHEMBL12944477 0.77 PABPC1 (0.44) HTR1AADRA1DADRA1AADRA1B
SCHEMBL1768196 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496578-A2 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME University of Notre Dame du Lac (US) 2012-09-12 EP claimed
US-20120220457-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME DOW AGROSCIENCES LLC (US) 2012-08-30 US claimed
WO-2011057145-A2 IMIDAZO[1,2-A] PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2011-05-12 WO claimed
EP-2875029-B1 5,5-HETEROAROMATIC ANTI-INFECTIVE COMPOUNDS MORASKI GARRETT (US) 2021-11-10 EP disclosed
US-10913737-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2021-02-09 US disclosed
US-20210009583-A1 DEUTERATED IMIDAZOPYRIDINES UNIVERSITY OF NOTRE DAME DU LAC (US) 2021-01-14 US disclosed
WO-2019175737-A1 DEUTERATED IMIDAZOPYRIDINES UNIVERSITY OF NOTRE DAME DU LAC (US) 2019-09-19 WO disclosed
US-20180354944-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2018-12-13 US disclosed
US-9908876-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2018-03-06 US disclosed
EP-3257854-A1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME University of Notre Dame du Lac (US) 2017-12-20 EP disclosed
US-9605002-B2 5,5-heteroaromatic anti-infective compounds UNIVERSITY OF NOTRE DAME DU LAC (US) 2017-03-28 US disclosed
US-9309238-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2016-04-12 US disclosed
US-20150210715-A1 5,5-HETEROAROMATIC ANTI-INFECTIVE COMPOUNDS UNIVERSITY OF NOTRE DAME DU LAC 2015-07-30 US disclosed
EP-2875029-A2 5,5-HETEROAROMATIC ANTI-INFECTIVE COMPOUNDS Moraski, Garrett (US) 2015-05-27 EP disclosed
WO-2014015167-A2 5,5-HETEROAROMATIC ANTI-INFECTIVE COMPOUNDS UNIVERSITY OF NOTRE DAME DU LAC (US) 2014-01-23 WO disclosed
EP-2496578-A2 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME University of Notre Dame du Lac (US) 2012-09-12 EP disclosed
US-20120220457-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME DOW AGROSCIENCES LLC (US) 2012-08-30 US disclosed
EP-2380886-A1 Process for the preparation of 2-aminosubstituted 1,3-benzothiazine-4-ones Makarov Vadim A. (RU) 2011-10-26 EP disclosed
WO-2011057145-A2 IMIDAZO[1,2-A] PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2011-05-12 WO disclosed
US-20070173570-A1 N-alkoxy-4, 4-dioxy-polyalkyl-piperidine compounds, with glycidyl or alkylcarbonyl groups as functional initiators for controlled radical polymerization FUSO FRANCESCO 2007-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10913737-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same RIF1, PYCR1, PNMT HTR1A 1992/4885ADRA1D 989/4885ADRA1A 1814/4885
US-20070173570-A1 N-alkoxy-4, 4-dioxy-polyalkyl-piperidine compounds, with glycidyl or alkylcarbonyl groups as functional initiators for controlled radical polymerization PTGER4, ALKBH3, PIGO HTR1A 1859/4885ADRA1D 2074/4885ADRA1A 3056/4885
US-20120220457-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME RIF1, PYCR1, PNMT HTR1A 1992/4885ADRA1D 989/4885ADRA1A 1814/4885
US-20210009583-A1 DEUTERATED IMIDAZOPYRIDINES SDHA, PDF, IDH2 HTR1A 4136/4885ADRA1D 1266/4885ADRA1A 2276/4885
US-20180354944-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME RIF1, PYCR1, PNMT HTR1A 1992/4885ADRA1D 989/4885ADRA1A 1814/4885
US-20150210715-A1 5,5-HETEROAROMATIC ANTI-INFECTIVE COMPOUNDS API5, CASP5, IL5 HTR1A 2842/4885ADRA1D 2313/4885ADRA1A 2022/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.