SCHEMBL1768256

SCHEMBL1768256

[NH]Cc1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.46
EPHX2 P34913 2/20 0.46
SOS1 Q07889 1/20 0.44
HSPB1 P04792 1/20 0.44
MAOB P27338 6/20 0.42
APP P05067 1/20 0.42
IDO1 P14902 3/20 0.41
AGXT P21549 2/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
ST14 Q9Y5Y6 1/20 0.40
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40
SCN4A P35499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL422167 0.85
SCHEMBL7367702 0.83 SOS1 (0.56) LTA4HEPHX2SOS1HSPB1SCN4A
SCHEMBL6289867 0.80 SOS1 (0.58) LTA4HEPHX2SOS1HSPB1SCN4A
SCHEMBL6290683 0.80 SOS1 (0.58) LTA4HEPHX2SOS1HSPB1SCN4A
SCHEMBL351854 0.80 SOS1 (0.58) LTA4HEPHX2SOS1HSPB1SCN4A
SCHEMBL1350555 0.79 LTA4H (0.61) LTA4HMAOA
SCHEMBL5563797 0.78 LTA4H (0.47) LTA4HEPHX2SOS1HSPB1MAOB
SCHEMBL919783 0.77 LOXL2 (0.73) LTA4HEPHX2SOS1MAOBIDO1
SCHEMBL6161106 0.77 LTA4H (0.65) LTA4HEPHX2SOS1HSPB1MAOB
SCHEMBL9106789 0.77 LTA4H (0.46) LTA4HEPHX2SOS1HSPB1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496578-A2 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME University of Notre Dame du Lac (US) 2012-09-12 EP claimed
US-20120220457-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME DOW AGROSCIENCES LLC (US) 2012-08-30 US claimed
WO-2011057145-A2 IMIDAZO[1,2-A] PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2011-05-12 WO claimed
US-10913737-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2021-02-09 US disclosed
US-20180354944-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2018-12-13 US disclosed
US-9908876-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2018-03-06 US disclosed
EP-3257854-A1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME University of Notre Dame du Lac (US) 2017-12-20 EP disclosed
US-20160318925-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2016-11-03 US disclosed
US-9309238-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same UNIVERSITY OF NOTRE DAME DU LAC (US) 2016-04-12 US disclosed
EP-2496578-A2 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME University of Notre Dame du Lac (US) 2012-09-12 EP disclosed
US-20120220457-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME DOW AGROSCIENCES LLC (US) 2012-08-30 US disclosed
WO-2011057145-A2 IMIDAZO[1,2-A] PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME UNIVERSITY OF NOTRE DAME DU LAC (US) 2011-05-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10913737-B2 Imidazo [1,2-a]pyridine compounds, synthesis thereof, and methods of using same RIF1, PYCR1, PNMT LTA4H 2150/4885EPHX2 2552/4885SOS1 3113/4885
US-20160318925-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME RIF1, PYCR1, PNMT LTA4H 2150/4885EPHX2 2552/4885SOS1 3113/4885
US-20120220457-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME RIF1, PYCR1, PNMT LTA4H 2150/4885EPHX2 2552/4885SOS1 3113/4885
US-20180354944-A1 IMIDAZO [1,2-a]PYRIDINE COMPOUNDS, SYNTHESIS THEREOF, AND METHODS OF USING SAME RIF1, PYCR1, PNMT LTA4H 2150/4885EPHX2 2552/4885SOS1 3113/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.