SCHEMBL1769121

SCHEMBL1769121

COC(=O)CN=Cc1ccc(OC)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.58
POLB P06746 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
CYP1A2 P05177 2/20 0.55
GSK3B P49841 1/20 0.51
CYP2C19 P33261 1/20 0.50
MAPT P10636 2/20 0.48
ALDH1A1 P00352 2/20 0.48
RAB9A P51151 2/20 0.48
KDM4E B2RXH2 1/20 0.48
GAA P10253 1/20 0.48
NPC1 O15118 1/20 0.48
HDAC3 O15379 2/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC10 Q969S8 1/20 0.48
GFER P55789 1/20 0.48
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23345343 1.00 KMT2A (0.58) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL1769120 1.00 KMT2A (0.58) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL11928783 0.87 CYP1A2 (0.53) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL6117540 0.87 CYP1A2 (0.53) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL6117537 0.87 CYP1A2 (0.53) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL23345327 0.86 HTT (0.51) KMT2APOLBSMN1; SMN2MAPTALDH1A1
SCHEMBL1769027 0.85 CYP1A2 (0.57) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL23326817 0.85 CYP1A2 (0.57) KMT2APOLBSMN1; SMN2CYP1A2GSK3B
SCHEMBL28360448 0.85 LMNA (0.45) KMT2APOLBSMN1; SMN2CYP1A2MAPT
SCHEMBL1769024 0.85 CYP1A2 (0.57) KMT2APOLBSMN1; SMN2CYP1A2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4582427-A1 USP1 INHIBITOR Shanghai Qilu Pharmaceutical Research and Development Centre Ltd. (CN) 2025-07-09 EP disclosed
CN-110577485-B Norcamphor derived [2, 1] -bridged ring ketene compounds and synthesis method and application thereof 武汉大学 2022-11-04 CN disclosed
CN-115108938-A Chiral alpha-substituted deuterated amino acid compound and preparation method thereof 武汉大学 2022-09-27 CN disclosed
CN-114940661-A Norcamphor derived [2,2,1] -bridged ketene compounds and synthesis method and application thereof 武汉大学 2022-08-26 CN disclosed
CN-114349585-A Catalytic asymmetric synthesis method and application of chiral alpha-deuterated pyrrolidine compound 武汉大学 2022-04-15 CN disclosed
CN-110577485-A Norcamphor derived [2,2,1] -bridged ketene compounds and synthesis method and application thereof 武汉大学 2019-12-17 CN disclosed
CN-106478645-A A kind of fragrant cyclosubstituted spiro indole diketopiperazine compound and its synthetic method 陕西科技大学 2017-03-08 CN disclosed
US-9321769-B2 Heterocyclic acrylamides and their use as pharmaceuticals FAB PHARMA S.A.S. (FR) 2016-04-26 US disclosed
US-20150232466-A1 NOVEL HETEROCYCLIC ACRYLAMIDES AND THEIR USE AS PHARMACEUTICALS FAB PHARMA S.A.S. (FR) 2015-08-20 US disclosed
US-9051321-B2 Heterocyclic acrylamides and their use as pharmaceuticals FAB PHARMA S.A.S. (FR) 2015-06-09 US disclosed
EP-2501693-A1 NOVEL HETEROCYCLIC ACRYLAMIDES AND THEIR USE AS PHARMACEUTICALS FAB Pharma SAS (FR) 2012-09-26 EP disclosed
US-8034810-B2 Matrix metalloproteinase inhibitors; antiinflammatory agengs; rheumatoid arthritis, osteoarthritis; antitumor, anticarcinogenic, and antimetastasis agents; respiratory system disorders, chronic obstructive pulmonary disease, deblocking, deprotecting NOVARTIS AG (CH) 2011-10-11 US disclosed
WO-2011061214-A1 NOVEL HETEROCYCLIC ACRYLAMIDES AND THEIR USE AS PHARMACEUTICALS FAB PHARMA SAS (FR) 2011-05-26 WO disclosed
EP-1202961-B1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES NOVARTIS AG (CH) 2010-01-20 EP disclosed
EP-2085379-A1 Arylsulfonamido-substituted hydroxamic acid derivatives Novartis AG (CH) 2009-08-05 EP disclosed
US-20080275127-A1 Arylsulfonamido-substituted hydroxamic acid derivatives BREITENSTEIN WERNER 2008-11-06 US disclosed
US-7138432-B1 Arylsulfonamido-substituted hydroxamic acid derivatives NOVARTIS AG (CH) 2006-11-21 US disclosed
EP-1202961-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES Novartis AG (CH) 2002-05-08 EP disclosed
WO-2001010827-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES NOVARTIS AG (CH) 2001-02-15 WO disclosed
US-5569661-A Process for the production of b-carbolines SCHERING AKTIENGESELLSCHAFT (DE) 1996-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150232466-A1 NOVEL HETEROCYCLIC ACRYLAMIDES AND THEIR USE AS PHARMACEUTICALS ACR, AADAC, AAAS KMT2A 4479/4885POLB 2880/4885SMN1; SMN2 4165/4885
US-20080275127-A1 Arylsulfonamido-substituted hydroxamic acid derivatives MMP13, MMP2, MMP1 KMT2A 2171/4885POLB 1365/4885SMN1; SMN2 4344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.