SCHEMBL17779981

SCHEMBL17779981

COc1ccc(C(=O)C(=O)C2CC2)cc1-c1cccc(C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P4HB P07237 2/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.43
BACE1 P56817 1/20 0.43
BCL9 O00512 2/20 0.43
CTNNB1 P35222 2/20 0.43
PDE4D Q08499 4/20 0.42
CTSA P10619 1/20 0.41
KDM1A O60341 1/20 0.41
USP30 Q70CQ3 1/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
HPSE Q9Y251 1/20 0.39
KIT P10721 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16109144 0.83 FFAR2 (0.46) PDE4DCTSA
SCHEMBL16108140 0.81 PAX8 (0.47) PDE4DUSP30
SCHEMBL16111924 0.78 MKNK1 (0.56) HPSECYP1A2CYP3A4
SCHEMBL7603613 0.77 RARA (0.55) P4HBPTGDR2PDE4DCTSAHPSE
SCHEMBL28788990 0.75 ROCK2 (0.51) P4HBPTGDR2ROCK2ROCK1HPSE
SCHEMBL16108312 0.75 KAT6A (0.44) USP30
SCHEMBL9469524 0.73 HTR7 (0.55) PDE4DKITCYP1A2CYP3A4CYP2D6
SCHEMBL1812722 0.73 KDM1A (0.49) PTGDR2BACE1PDE4DCTSAKDM1A
SCHEMBL4974725 0.73 AR (0.52) PTGDR2BACE1PDE4DCTSAKDM1A
SCHEMBL1811323 0.72 LPAR1 (0.51) PTGDR2BCL9CTNNB1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9353089-B2 Compositions and methods for the treatment of malaria SAINT LOUIS UNIVERSITY (US) 2016-05-31 US disclosed