SCHEMBL17786111

SCHEMBL17786111

CS(=O)(=O)c1ccc(C(N)=O)c(N)c1C1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.38
CDC7 O00311 1/20 0.38
IKBKB O14920 2/20 0.37
CHUK O15111 2/20 0.37
PARP2 Q9UGN5 3/20 0.34
PLAT P00750 1/20 0.34
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
HTR6 P50406 1/20 0.33
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2466003 0.82 CDC7 (0.36) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL4446215 0.77 QDPR (0.48) PARP1CDC7IKBKBCHUKPARP2
Hydrochloric Acid SCHEMBL4435861 0.76 QDPR (0.47) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL4560312 0.75 PARP1 (0.38) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL17786119 0.74 IKBKB (0.47) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL6233771 0.73 PARP1 (0.36) PARP1CDC7IKBKBCHUKTLR8
SCHEMBL8498415 0.71 LMNA (0.37) PARP1PARP2HTR6
SCHEMBL5808501 0.71 HTR2C (0.44) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL28325510 0.70 PARP1 (0.57) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL2465997 0.70 SYK (0.43) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016086153-A2 USE OF TETRAHYDRO!NDAZOLYLBEIMZAMIDE AND TETRAHYDROINDOLYLBENZAMIDE DERIVATIVES FOR THE TREATMENT OF HUMAN IMMUNODEFICIENCY VIRUS (HIV) AND ACQUIRED IMMUNE DEFICIENCY SYNDROME (AIDS) ESANEX, INC. (US) 2016-06-02 WO disclosed