SCHEMBL28547235

SCHEMBL28547235

CCNc1c(N)n(Cc2ccc(Cl)cc2)c(S)nc1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 4/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TYMS P04818 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
CYP2C19 P33261 1/20 0.39
CASP7 P55210 1/20 0.39
HIF1A Q16665 1/20 0.39
TLR7 Q9NYK1 6/20 0.38
TLR8 Q9NR97 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814738 0.81 TNF (0.42) RAB9AALDH1A1KDM4EHSD17B10HPGD
SCHEMBL28555375 0.80 RAB9A (0.40) RAB9AALDH1A1KDM4EHSD17B10MEN1
SCHEMBL17814737 0.76 ALDH1A1 (0.41) RAB9AALDH1A1KDM4EHSD17B10HPGD
SCHEMBL17814735 0.68 PNP (0.57) KMT2ATLR7TLR8NPC1
SCHEMBL30804819 0.68 BRD4 (0.42) RAB9AALDH1A1KDM4EHSD17B10HPGD
SCHEMBL28537635 0.68 TSHR (0.37) RAB9AALDH1A1KDM4EHSD17B10HPGD
SCHEMBL29172435 0.67 P2RX3 (0.42) LMNANOD1BRD4GAA
SCHEMBL28538573 0.63 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL21389540 0.62 BRD4 (0.62) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL21389574 0.62 BRD4 (0.62) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed