SCHEMBL178204

SCHEMBL178204

Nc1nc(-c2ccc(Cl)cc2)c(C(=O)c2cccc(F)c2)s1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 6/20 0.58
CDK5R1 Q15078 6/20 0.58
RORB Q92753 10/20 0.51
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
RORC P51449 2/20 0.46
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10092890 0.89 RORB (0.65) CDK5CDK5R1RORBCCNA2CDK2
SCHEMBL257393 0.89 RORB (0.60) CDK5CDK5R1RORBCCNA2CDK2
SCHEMBL178218 0.85 ADORA3 (0.60) RORBRORCADORA3ADORA2AADORA1
SCHEMBL257438 0.83 ADORA3 (0.54) RORBRORCADORA3ADORA2AADORA1
SCHEMBL10092883 0.81 RORB (0.67) RORBCCNA2CDK2RORCADORA3
SCHEMBL168526 0.81 RORB (0.70) RORBCCNA2CDK2RORCADORA1
SCHEMBL257615 0.80 RORB (0.72) RORBCCNA2CDK2RORCADORA2A
SCHEMBL257616 0.80 ADORA3 (0.64) RORBADORA3ADORA2AADORA1
SCHEMBL10092885 0.79 RORB (0.70) RORBRORCADORA3ADORA2AADORA1
SCHEMBL257436 0.79 RORB (0.66) RORBRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed