SCHEMBL178218

SCHEMBL178218

Nc1nc(-c2ccc(Cl)cc2)c(C(=O)c2ccccc2)s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.60
ADORA1 P30542 2/20 0.60
ADORA2A P29274 1/20 0.60
LMNA P02545 3/20 0.55
NPSR1 Q6W5P4 3/20 0.55
RORB Q92753 6/20 0.54
SMN1; SMN2 Q16637 3/20 0.53
ALDH1A1 P00352 2/20 0.53
MAPT P10636 2/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
ADORA2B P29275 1/20 0.51
POLB P06746 1/20 0.50
HSD17B10 Q99714 1/20 0.50
RORC P51449 2/20 0.49
NPC1 O15118 1/20 0.49
NFKB1 P19838 1/20 0.49
PPARG P37231 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257616 0.94 ADORA3 (0.64) ADORA3ADORA1ADORA2ALMNANPSR1
SCHEMBL257438 0.93 ADORA3 (0.54) ADORA3ADORA1ADORA2ALMNANPSR1
SCHEMBL165773 0.90 ADORA3 (0.61) ADORA3ADORA1ADORA2ALMNANPSR1
SCHEMBL257393 0.88 RORB (0.60) ADORA3ADORA1ADORA2ALMNANPSR1
SCHEMBL10092883 0.85 RORB (0.67) ADORA3ADORA1ADORA2ARORBALDH1A1
SCHEMBL257432 0.85 RORB (0.74) ADORA3ADORA1ADORA2ALMNANPSR1
SCHEMBL178204 0.85 CDK5 (0.58) ADORA3ADORA1ADORA2ARORBPOLB
SCHEMBL257437 0.84 RORB (0.76) RORBSMN1; SMN2ALDH1A1MAPTMEN1
SCHEMBL10092885 0.83 RORB (0.70) ADORA3ADORA1ADORA2ALMNANPSR1
SCHEMBL27653923 0.82 ALDH1A1 (0.64) ADORA3NPSR1RORBSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed