SCHEMBL17844168

SCHEMBL17844168

COCCn1sc(-c2ccccc2)c(NC2CCOCC2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.37
MAPK14 Q16539 5/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ADORA2B P29275 1/20 0.34
PDE4B Q07343 5/20 0.34
LCK P06239 1/20 0.34
PDE7A Q13946 1/20 0.34
POLB P06746 1/20 0.33
BRD4 O60885 1/20 0.33
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844156 0.87 ADORA2B (0.36) MAPK14ALDH1A1CYP1A2CASP1CASP7
SCHEMBL5199815 0.85 ADORA2B (0.35) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL17844144 0.74 FAAH (0.40) MAPK1ALDH1A1CYP1A2CASP1CASP7
SCHEMBL17844251 0.73 FAAH (0.39) ALDH1A1ADORA2BPDE4BPDE7APOLB
SCHEMBL2001680 0.70 MAPK1 (0.39) MAPK1MAPK14ALDH1A1CYP1A2CASP1
SCHEMBL3503724 0.70 MAPT (0.45) MAPK1ALDH1A1CYP1A2HSD17B10
SCHEMBL17844132 0.69 FAAH (0.39) ALDH1A1HSD17B10ADORA2B
SCHEMBL5186704 0.67 FAAH (0.38) ALDH1A1HSD17B10ADORA2BPDE4BPDE7A
SCHEMBL17844164 0.65 KAT2B (0.38) MAPK1CYP1A2POLB
SCHEMBL5185885 0.65 LMNA (0.43) MAPK1ALDH1A1CYP1A2HSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100619-A2 TREATMENT AND DIAGNOSIS OF CANCER RGENIX, INC. (US) 2016-06-23 WO disclosed