SCHEMBL17845490

SCHEMBL17845490

COc1cccc(NC2CCO[C]2N)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.49
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 1/20 0.45
STAT1 P42224 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
PKM P14618 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845615 0.84 ROCK2 (0.46) ROCK2NPC1RAB9AL3MBTL1ALDH1A1
SCHEMBL17845583 0.84 ROCK2 (0.46) ROCK2NPC1RAB9AL3MBTL1ALDH1A1
SCHEMBL17845604 0.82 GAA (0.47) NPC1RAB9AL3MBTL1ALDH1A1MEN1
SCHEMBL17845650 0.79 FADS1 (0.50) NPC1RAB9AALDH1A1LMNAMEN1
SCHEMBL17845575 0.79 KDM4E (0.43) ROCK2NPC1RAB9AMEN1KMT2A
SCHEMBL17845573 0.79 KMT2A (0.39) NPC1ALDH1A1MEN1KMT2ACYP3A4
SCHEMBL1298275 0.75 ALDH1A1 (0.54) ROCK2NPC1RAB9AALDH1A1LMNA
SCHEMBL29724427 0.75 ALDH1A1 (0.54) ROCK2NPC1RAB9AALDH1A1LMNA
SCHEMBL2481941 0.72 NPC1 (0.57) ROCK2NPC1RAB9AALDH1A1LMNA
SCHEMBL17845540 0.71 RAB9A (0.43) ROCK2NPC1RAB9AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233860-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS Univerzita Palackého V Olomouci (CZ) 2017-10-25 EP disclosed
WO-2016095881-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-06-23 WO disclosed