SCHEMBL17845604

SCHEMBL17845604

COc1ccc(NC2CCO[C]2N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.47
TSHR P16473 1/20 0.47
MAPT P10636 5/20 0.46
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 2/20 0.46
NR4A1 P22736 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MAPK1 P28482 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
THRB P10828 1/20 0.41
RECQL P46063 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HPGD P15428 1/20 0.40
ENPP2 Q13822 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845700 0.83 GAA (0.46) GAATSHRMAPTALDH1A1SMN1; SMN2
SCHEMBL17845446 0.83 GAA (0.46) GAATSHRMAPTALDH1A1SMN1; SMN2
SCHEMBL17845490 0.82 ROCK2 (0.49) MAPTALDH1A1NPC1RAB9AMAPK1
SCHEMBL17845466 0.76 ALDH1A1 (0.42) GAAALDH1A1SMN1; SMN2KDM4ENPC1
SCHEMBL2563095 0.71 ALDH1A1 (0.55) GAATSHRMAPTALDH1A1SMN1; SMN2
SCHEMBL17845573 0.69 KMT2A (0.39) TSHRALDH1A1SMN1; SMN2NPC1TDP1
SCHEMBL17845650 0.69 FADS1 (0.50) TSHRMAPTALDH1A1NPC1RAB9A
SCHEMBL17845575 0.69 KDM4E (0.43) GAASMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL3108892 0.68 RAB9A (0.57) GAAMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL17845717 0.68 MAPK1 (0.39) GAATSHRMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233860-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS Univerzita Palackého V Olomouci (CZ) 2017-10-25 EP disclosed
WO-2016095881-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-06-23 WO disclosed