SCHEMBL17845532

SCHEMBL17845532

CCOc1cccc(NC2CCO[C]2F)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.42
SYK P43405 1/20 0.42
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 2/20 0.39
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
PLAU P00749 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845615 0.85 ROCK2 (0.46) ROCK2RAB9ANPC1KMT2AMEN1
SCHEMBL17845449 0.85 ROCK2 (0.42) ROCK2SYKRAB9ANPC1HTT
SCHEMBL17845602 0.78 KDM4E (0.44) ROCK2RAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL17845716 0.75 FADS1 (0.50) RAB9ANPC1HTTSMN1; SMN2KMT2A
SCHEMBL17845542 0.74 DDB1 (0.40) HTTSMN1; SMN2ALDH1A1
SCHEMBL17845550 0.72 SYK (0.38) ROCK2SYKRAB9ANPC1HTT
SCHEMBL17845490 0.70 ROCK2 (0.49) ROCK2RAB9ANPC1KMT2AMEN1
SCHEMBL17845768 0.70 HTT (0.38) ROCK2SYKRAB9ANPC1HTT
SCHEMBL17845583 0.69 ROCK2 (0.46) ROCK2RAB9ANPC1KMT2AMEN1
SCHEMBL18164614 0.69 SMN1; SMN2 (0.44) ROCK2SYKRAB9ANPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233860-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS Univerzita Palackého V Olomouci (CZ) 2017-10-25 EP disclosed
WO-2016095881-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-06-23 WO disclosed