SCHEMBL17845569

SCHEMBL17845569

Fc1ccc(NC2CCO[C]2Cl)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
POLB P06746 1/20 0.37
ROCK2 O75116 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 2/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
P2RX7 Q99572 2/20 0.35
MAPK14 Q16539 2/20 0.34
MAPK8 P45983 1/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845712 0.84 KMT2A (0.33) ROCK2KMT2A
SCHEMBL17845530 0.81 GAA (0.41) GAANPC1RAB9APOLBKMT2A
SCHEMBL17845762 0.80 EPHX2 (0.36) KMT2ALMNAP2RX7TAS1R3TAS1R1
SCHEMBL17845595 0.78 DDB1 (0.43) NPC1RAB9APOLBLMNAP2RX7
SCHEMBL17845386 0.76 ROCK2 (0.36) GAAROCK2P2RX7TP53
SCHEMBL17845497 0.76 KDM4E (0.43) GAANPC1RAB9AROCK2KMT2A
SCHEMBL17845706 0.75 RAB9A (0.40) NPC1RAB9AHTTKMT2ALMNA
SCHEMBL17845726 0.71 KMT2A (0.40) GAANPC1RAB9AKMT2APKM
SCHEMBL17845703 0.70 ESR1 (0.32)
SCHEMBL17845720 0.69 NPC1 (0.34) GAANPC1RAB9APOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233860-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS Univerzita Palackého V Olomouci (CZ) 2017-10-25 EP disclosed
WO-2016095881-A1 SUBSTITUTED 6-ANILINO-9-HETEROCYCLYLPURINE DERIVATIVES FOR INHIBITION OF PLANT STRESS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-06-23 WO disclosed