SCHEMBL1785215

SCHEMBL1785215

O=C(O)c1cc(-n2cccc2)ccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.62
POLB P06746 5/20 0.62
KDM4E B2RXH2 3/20 0.62
HPGD P15428 1/20 0.62
MAPK1 P28482 1/20 0.62
HSD17B10 Q99714 1/20 0.62
TDP1 Q9NUW8 4/20 0.58
CTSB P07858 1/20 0.58
TP53 P04637 1/20 0.53
L3MBTL1 Q9Y468 3/20 0.51
MRGPRX4 Q96LA9 1/20 0.49
SERPINE1 P05121 2/20 0.49
CASP6 P55212 3/20 0.48
CTDSP1 Q9GZU7 3/20 0.48
KMT2A Q03164 2/20 0.48
NSD2 O96028 2/20 0.48
ALK Q9UM73 1/20 0.48
PKM P14618 1/20 0.48
APEX1 P27695 1/20 0.48
CASP3 P42574 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3140547 0.86 ALDH1A1 (0.67) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL1788237 0.84 ALDH1A1 (0.59) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL2757862 0.81 KMT2A (0.65) ALDH1A1POLBKDM4EHPGDTDP1
SCHEMBL130491 0.80 KDM4E (0.74) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL1786657 0.79 POLB (0.62) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL15714465 0.76 ALDH1A1 (1.00) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL5323825 0.75 ALDH1A1 (0.57) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL28034614 0.74 MAPT (0.51) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL15123245 0.74 IP6K1 (0.66) ALDH1A1POLBKDM4EHPGDMAPK1
SCHEMBL3045754 0.74 ALDH1A1 (0.73) ALDH1A1POLBKDM4EHPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12497643-B2 Endo-S2 mutants as glycosynthases, method of making and use for glycoengineering of glycoproteins UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2025-12-16 US disclosed
US-12187662-B2 FOXM1 inhibitor compositions and methods of using the same THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2025-01-07 US disclosed
US-20240216345-A1 NEW METHOD FOR TREATING DENGUE VIRUS INFECTION INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2024-07-04 US disclosed
US-11845970-B2 Endo-S2 mutants as glycosynthases, method of making and use for glycoengineering of glycoproteins UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2023-12-19 US disclosed
EP-3402815-B1 ENDO-S2 MUTANTS AS GLYCOSYNTHASES, METHOD OF MAKING AND USE FOR GLYCOENGINEERING OF GLYCOPROTEINS UNIV MARYLAND (US) 2023-12-06 EP disclosed
US-20230348947-A1 ENDO-S2 MUTANTS AS GLYCOSYNTHASES, METHOD OF MAKING AND USE FOR GLYCOENGINEERING OF GLYCOPROTEINS UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2023-11-02 US disclosed
US-20230313325-A1 METHODS FOR DETECTION OF PATHOGENIC INFECTIONS USING RED BLOOD CELL-CONTAINING PATIENT SAMPLES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2023-10-05 US disclosed
US-11643450-B2 Chemoenzymatic glycoengineering of antibodies and Fc fragments thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-05-09 US disclosed
EP-4146820-A1 METHODS FOR DETECTION OF PATHOGENIC INFECTIONS USING RED BLOOD CELL-CONTAINING PATIENT SAMPLES The Trustees of The University of Pennsylvania (US) 2023-03-15 EP disclosed
EP-2812442-B9 CHEMOENZYMATIC GLYCOENGINEERING OF ANTIBODIES AND FC FRAGMENTS THEREOF UNIV MARYLAND (US) 2023-02-15 EP disclosed
EP-2607357-A1 BENZOTHIAZOLES AS GHRELIN RECEPTOR MODULATORS Astrazeneca AB (SE) 2013-06-26 EP disclosed
US-20120115845-A1 THERAPEUTIC AGENTS ALLEN JACK MCQUEEN (GB) 2012-05-10 US disclosed
US-20110124621-A1 BENZOTHIAZOLES AS GHRELIN RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2011-05-26 US disclosed
CN-101883762-A Benzothiazoles as modulators of growth hormone releasing hormone receptors ASTRAZENECA AB 2010-11-10 CN disclosed
EP-2205576-A1 BENZOTHIAZOLES AS GHRELIN RECEPTOR MODULATORS AstraZeneca AB (SE) 2010-07-14 EP disclosed
US-20090186870-A1 Therapeutic Agents - 802 ASTRAZENECA AB (SE) 2009-07-23 US disclosed
WO-2009047558-A1 BENZOTHIAZOLES AS GHRELIN RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2009-04-16 WO disclosed
US-20080039428-A1 Antiretroviral combination therapy PANACOS PHARMACEUTICALS, INC. (US) 2008-02-14 US disclosed
US-20070232684-A1 Compounds for inhibition of HIV infection by blocking HIV entry NEW YORK BLOOD CENTER 2007-10-04 US disclosed
US-7241803-B2 Compounds for inhibition of HIV infection by blocking HIV entry NEW YORK BLOOD CENTER (US) 2007-07-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232684-A1 Compounds for inhibition of HIV infection by blocking HIV entry SDF4, NUCB2, CXCR4 ALDH1A1 4651/4885POLB 3253/4885KDM4E 4676/4885
US-20120115845-A1 THERAPEUTIC AGENTS GPR119, MC2R, MC4R ALDH1A1 650/4885POLB 4524/4885KDM4E 3215/4885
US-20090186870-A1 Therapeutic Agents - 802 GPR119, SLC5A2, MC2R ALDH1A1 918/4885POLB 3987/4885KDM4E 3524/4885
US-20110124621-A1 BENZOTHIAZOLES AS GHRELIN RECEPTOR MODULATORS GPR119, GHSR, GLP1R ALDH1A1 2084/4885POLB 4687/4885KDM4E 1188/4885
US-12187662-B2 FOXM1 inhibitor compositions and methods of using the same FOXM1, FOXO1, TP53 ALDH1A1 2437/4885POLB 356/4885KDM4E 495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.