SCHEMBL18023968

SCHEMBL18023968

N#Cc1ccc(C(=O)Nc2c(Cl)cc(C(F)(c3ccc(Cl)cc3)C(F)(F)F)cc2Cl)cc1NO

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
S1PR3 Q99500 13/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
S1PR1 P21453 5/20 0.39
AR P10275 2/20 0.37
S1PR2 O95136 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16330798 0.87 S1PR3 (0.52) S1PR3S1PR1S1PR2
SCHEMBL12437132 0.87 S1PR3 (0.40) S1PR3CYP1A2CYP2D6CYP2C19RAB9A
SCHEMBL12438374 0.86 S1PR3 (0.39) HDAC1HDAC8HDAC6S1PR3CYP1A2
SCHEMBL12437133 0.85 TAS1R3 (0.40) HDAC1HDAC8HDAC6S1PR3CYP1A2
SCHEMBL14120380 0.85 TRPV1 (0.46) HDAC1HDAC8HDAC6S1PR3RAB9A
SCHEMBL12437616 0.85 ALDH1A1 (0.46) S1PR3RAB9AS1PR1MEN1KMT2A
SCHEMBL12437620 0.84 MEN1 (0.46) HDAC1HDAC8HDAC6S1PR3CYP1A2
SCHEMBL12437547 0.83 S1PR3 (0.43) S1PR3S1PR1ARMEN1KMT2A
SCHEMBL14120559 0.83 LMNA (0.48) S1PR3S1PR1MEN1KMT2A
SCHEMBL9894400 0.75 S1PR3 (0.47) S1PR3S1PR1ARS1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531484-B1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2016-08-17 EP disclosed