SCHEMBL1811550

SCHEMBL1811550

FC(F)(F)c1ccc(C2CCNC2)cc1

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.79
HTR3A P46098 1/20 0.59
P2RY14 Q15391 1/20 0.53
TMEM97 Q5BJF2 1/20 0.53
HTR2A P28223 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17938547 1.00 HTR2C (0.79) HTR2CHTR3AP2RY14TMEM97HTR2A
SCHEMBL16660400 1.00 HTR2C (0.79) HTR2CHTR3AP2RY14TMEM97HTR2A
Hydrochloric Acid SCHEMBL4573167 0.98 HTR2C (0.80) HTR2CHTR3AP2RY14TMEM97HTR2A
SCHEMBL12809959 0.91 HTR2C (0.66) HTR2CHTR3AHTR2A
Oxalic Acid SCHEMBL3543097 0.91 HTR2C (0.66) HTR2CHTR3AP2RY14TMEM97
Hydrochloric Acid SCHEMBL568208 0.89 HTR2C (0.67) HTR2CHTR3AHTR2A
Trifluoroacetic Acid SCHEMBL22638730 0.89 HTR2C (0.64) HTR2CHTR3AP2RY14TMEM97
SCHEMBL373310 0.89 HTR2C (1.00) HTR2CP2RY14TMEM97HTR2A
Hydrochloric Acid SCHEMBL381390 0.87 HTR2C (1.00) HTR2CP2RY14TMEM97HTR2A
SCHEMBL22778147 0.86 HTR2C (0.60) HTR2CP2RY14TMEM97HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119731162-A PRMT5 inhibitors 北京望实智慧科技有限公司 2025-03-28 CN disclosed
US-20230227428-A1 AMIDO COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2023-07-20 US disclosed
US-20230227428-A1 AMIDO COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2023-07-20 US disclosed
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-115698009-A CD73 inhibiting 2,4-dioxopyrimidine compounds 吉利德科学公司 2023-02-03 CN disclosed
WO-2021253098-A1 AMIDO COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2021-12-23 WO disclosed
WO-2021253098-A1 AMIDO COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2021-12-23 WO disclosed
WO-2021222522-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed
US-11046714-B2 2,2-difluorodioxolo A2A receptor antagonists MERCK SHARP & DOHME CORP. (US) 2021-06-29 US disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed
US-20070299071-A1 Substituted phenyl methanone derivatives F. HOFFMANN-LA ROCHE AG (CH) 2007-12-27 US disclosed
US-20070299071-A1 Substituted phenyl methanone derivatives F. HOFFMANN-LA ROCHE AG (CH) 2007-12-27 US disclosed
US-20070299071-A1 Substituted phenyl methanone derivatives F. HOFFMANN-LA ROCHE AG (CH) 2007-12-27 US disclosed
WO-2007147770-A2 SUBSTITUTED PHENYL METHANONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-12-27 WO disclosed
WO-2007147770-A2 SUBSTITUTED PHENYL METHANONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-12-27 WO disclosed
CN-101056845-A Substituted aniline derivatives LUNDBECK & CO AS H (DK) 2007-10-17 CN disclosed
CN-1150165-C 1-arylsulfonyl-2-aryl-pyrrolidine derivatives for the treatment of central nervous system disorders - 2004-05-19 CN disclosed
CN-1345311-A 1-arenesulfonyl-2-aryl-pyrolidine and piperidine derivatives for treatment of CNS disorders HOFFMANN LA ROCHE (CH) 2002-04-17 CN disclosed
US-5861416-A TREATMENT OF ASTHMA OR COUGH MERRELL PHARMACEUTICALS INC. (US) 1999-01-19 US disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227428-A1 AMIDO COMPOUNDS RIPK1, RIPK3, MLKL HTR2C 4642/4885HTR3A 3838/4885P2RY14 1619/4885
US-20070299071-A1 Substituted phenyl methanone derivatives CYP11B1, CYP11B2, MC2R HTR2C 70/4885HTR3A 72/4885P2RY14 1373/4885
US-11046714-B2 2,2-difluorodioxolo A2A receptor antagonists ADORA2A, ADORA2B, ADORA3 HTR2C 6/4885HTR3A 15/4885P2RY14 193/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.