SCHEMBL18138237

SCHEMBL18138237

CCn1cc(N=O)c(NC(=O)OC(C)(C)C)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.37
NPC1 O15118 4/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
GAA P10253 1/20 0.34
SCD O00767 1/20 0.34
RAB9A P51151 2/20 0.34
RECQL P46063 1/20 0.34
CYP17A1 P05093 1/20 0.34
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33
ACSS2 Q9NR19 1/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18138249 0.90 CNR2 (0.35) RORCNPC1ALDH1A1KDM4EPTGDR2
SCHEMBL18138239 0.84 DRD2 (0.39) ALDH1A1PTGDR2HDAC3HDAC8NCOR2
SCHEMBL18138297 0.79 GSK3B (0.33) NPC1PTGDR2HDAC3HDAC8NCOR2
SCHEMBL19026780 0.71 RAB9A (0.36) NPC1SMN1; SMN2RAB9ARECQLCYP17A1
SCHEMBL28055517 0.70 RAF1 (0.49) NPC1ALDH1A1PTGDR2SMN1; SMN2RAB9A
SCHEMBL24896677 0.69 L3MBTL1 (0.46) NPC1ALDH1A1KDM4EHDAC3HDAC8
SCHEMBL12764246 0.69 NPC1 (0.48) NPC1ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL28988125 0.68 HDAC3 (0.52) HDAC3HDAC8NCOR2SCDCYP17A1
SCHEMBL15885557 0.68 NPSR1 (0.54) NPC1ALDH1A1KDM4EPTGDR2LMNA
SCHEMBL16447788 0.67 PTGDR2 (0.40) KDM4EPTGDR2HDAC3HDAC8NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016164754-A1 FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2016-10-13 WO disclosed