SCHEMBL18154540

SCHEMBL18154540

O=c1oc2ccccc2c(-c2ccccc2)c1CCBr

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
NQO1 P15559 3/20 0.46
TP53 P04637 3/20 0.46
LMNA P02545 3/20 0.46
CYP3A4 P08684 2/20 0.46
TSHR P16473 2/20 0.46
MAPK1 P28482 2/20 0.46
MEN1 O00255 1/20 0.46
ABCB11 O95342 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.46
PDE4D Q08499 1/20 0.46
PCSK7 Q16549 1/20 0.46
GPR35 Q9HC97 1/20 0.46
MAPT P10636 2/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CYP19A1 P11511 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699860 0.89 NPC1 (0.48) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL18150080 0.88 TP53 (0.49) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL18154548 0.85 NQO1 (0.50) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL18150087 0.81 BRAF (0.53) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL28455189 0.77 ALDH1A1 (0.47) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL1800595 0.77 CA1 (0.56) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL9311 0.76 CA1 (0.56) ALDH1A1TP53LMNACYP3A4MAPK1
SCHEMBL28053823 0.76 CA1 (0.51) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL27594102 0.72 MAOA (0.50) ALDH1A1NQO1TP53LMNACYP3A4
SCHEMBL28859670 0.72 CA1 (0.51) ALDH1A1NQO1TP53LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3283481-A1 CHROMENE DERIVATIVES AS PHOSHOINOSITIDE 3-KINASES INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2018-02-21 EP disclosed
WO-2016166239-A1 CHROMENE DERIVATIVES AS PHOSHOINOSITIDE 3-KINASES INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2016-10-20 WO disclosed