SCHEMBL1826601

SCHEMBL1826601

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nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
SLC7A11 Q9UPY5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555854 0.78 GSR (0.43)
Cysteine SCHEMBL19359143 0.73 PTGS1 (0.52) PTGS1SLC7A11
Cysteine SCHEMBL19359142 0.73 PTGS1 (0.52) PTGS1SLC7A11
SCHEMBL28616609 0.71 KDM4E (0.30)
Cysteine SCHEMBL1889352 0.69 PTGS1 (0.46) PTGS1SLC7A11
SCHEMBL6022461 0.69
SCHEMBL11880209 0.69
SCHEMBL3794407 0.68 CASP3 (0.35) PTGS1
SCHEMBL8909319 0.68
Cysteine SCHEMBL16208953 0.66 PTGS1 (0.61) PTGS1SLC7A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023097222-A1 CELL DELIVERY COMPOSITIONS AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-01 WO claimed
EP-2987805-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2016-02-24 EP claimed
US-20150252093-A1 GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE ANALOGUES IPSEN PHARMA S.A.S. (FR) 2015-09-10 US claimed
US-20150175665-A1 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL IPSEN PHARMA S.A.S. (FR) 2015-06-25 US claimed
US-8999940-B2 Analogues of glucose-dependent insulinotropic polypeptide (GIP) modified at N-terminal IPSEN PHARMA S.A.S. (FR) 2015-04-07 US claimed
US-20110136725-A1 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL BIOMEASURE, INCORPORATED 2011-06-09 US claimed
EP-2328922-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2011-06-08 EP claimed
EP-2323678-A2 GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE ANALOGUES IPSEN PHARMA S.A.S. (FR) 2011-05-25 EP claimed
EP-2320923-A2 TRUNCATED ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2011-05-18 EP claimed
EP-2318433-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL IPSEN PHARMA S.A.S. (FR) 2011-05-11 EP claimed
WO-2010016940-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO claimed
WO-2010016935-A2 TRUNCATED ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO claimed
WO-2010016938-A2 GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE ANALOGUES IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO claimed
WO-2010016944-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO claimed
WO-2010016936-A1 PHARMACEUTICAL COMPOSITIONS OF ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO claimed
WO-2023097222-A1 CELL DELIVERY COMPOSITIONS AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-01 WO disclosed
EP-2323678-B1 GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE ANALOGUES IPSEN PHARMA SAS (FR) 2016-03-23 EP disclosed
WO-2010016940-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO disclosed
WO-2010016935-A2 TRUNCATED ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO disclosed
WO-2010016944-A2 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL IPSEN PHARMA S.A.S. (FR) 2010-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150252093-A1 GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE ANALOGUES GIPR, GPR119, GLP1R PTGS1 2005/4885SLC7A11 1213/4885
US-20150175665-A1 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL GIPR, GPR119, GLP1R PTGS1 2525/4885SLC7A11 1071/4885
US-20110136725-A1 ANALOGUES OF GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE (GIP) MODIFIED AT N-TERMINAL GIPR, GPR119, GLP1R PTGS1 2539/4885SLC7A11 1087/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.