SCHEMBL18280255

SCHEMBL18280255

NC(=O)c1ccc(OCC(=O)N(Cc2cc(Cl)ccc2Cl)c2cnccc2N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GLA P06280 1/20 0.38
KCNH2 Q12809 3/20 0.36
THRB P10828 1/20 0.35
PARP10 Q53GL7 2/20 0.35
AOC3 Q16853 1/20 0.35
SGMS2 Q8NHU3 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
MAP4K4 O95819 1/20 0.34
NR4A2 P43354 1/20 0.34
MAPT P10636 2/20 0.34
PARP15 Q460N3 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16796528 0.87 SGMS2 (0.41) CYP1A2CYP3A4CYP2C9CYP2C19GLA
SCHEMBL18148865 0.83 SLC6A2 (0.38) SGMS2
SCHEMBL18148861 0.77 TSPO (0.41) SGMS2MAPTLMNAGAA
SCHEMBL18280256 0.67 TP53 (0.44) PARP10NR4A2MAPTPARP15
SCHEMBL6232632 0.59 KMT2A (0.39) CYP1A2CYP3A4CYP2C19KCNH2SGMS2
SCHEMBL11099690 0.59 PARP10 (0.66) PARP10AOC3PARP15
SCHEMBL4638814 0.59 NR4A2 (0.62) PARP10NR4A2PARP15NPC1RAB9A
SCHEMBL30765129 0.58 NR4A2 (0.75) PARP10NR4A2MAPTPARP15NPC1
SCHEMBL16796529 0.58 KDM4C (0.44) GAA
SCHEMBL29718832 0.58 SIRT1 (0.47) CYP3A4SMN1; SMN2MAPTLMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080117-B1 IMIDAZOPYRIDINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB Biopharma SRL (BE) 2020-06-03 EP disclosed
US-9890154-B2 Imidazopyridine derivatives as modulators of TNF activity UCB BIOPHARMA SPRL (BE) 2018-02-13 US disclosed
US-20160355509-A1 Imidazopyridine Derivatives as Modulators of TNF Activity UCB BIOPHARMA SPRL (BE) 2016-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160355509-A1 Imidazopyridine Derivatives as Modulators of TNF Activity TNF, TNFRSF1A, TNFRSF9 CYP1A2 1265/4885CYP3A4 798/4885CYP2C9 1494/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.