SCHEMBL1831846

SCHEMBL1831846

CC(=O)NCC[N+](C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
MAPK1 P28482 2/20 0.52
HIF1A Q16665 1/20 0.52
TSHR P16473 1/20 0.48
ALDH1A1 P00352 1/20 0.46
PAOX Q6QHF9 3/20 0.43
ACHE P22303 2/20 0.42
ADRA1A P35348 2/20 0.41
CHRM5 P08912 3/20 0.41
CHRM1 P11229 3/20 0.41
CHRM3 P20309 3/20 0.41
CHRM2 P08172 2/20 0.41
CHRM4 P08173 2/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNA7 P36544 2/20 0.41
CHRNA4 P43681 2/20 0.41
PGR P06401 1/20 0.41
HTR1A P08908 1/20 0.41
TBXA2R P21731 1/20 0.41
CHRNB4 P30926 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8763339 0.85 KDM4E (0.61) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL14448326 0.84 KDM4E (0.52) KDM4EMAPK1HIF1ATSHRALDH1A1
Hydrochloric Acid SCHEMBL4058823 0.83 KDM4E (0.58) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL19192288 0.83 KDM4E (0.65) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL15473377 0.82 KDM4E (0.50) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL15470699 0.80 KDM4E (0.48) KDM4EMAPK1HIF1ATSHRALDH1A1
Hydrochloric Acid SCHEMBL1260787 0.77 LMNA (0.40) MAPK1TSHRALDH1A1ACHEADRA1A
SCHEMBL2694530 0.77 ACHE (0.37) KDM4EMAPK1ALDH1A1ACHEADRA1A
SCHEMBL16437514 0.77 KDM4E (0.44) KDM4EMAPK1HIF1ATSHRALDH1A1
SCHEMBL9547184 0.77 KDM4E (0.44) KDM4EMAPK1HIF1ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008044099-A1 CHARGE TRANSFER COMPLEXES IN THE TREATMENT OF INFLAMMATORY BOWEL DISEASES GHISALBERTI CARLO (BR) 2008-04-17 WO claimed
CN-116348084-A Cosmetic compositions, kits, and methods of making and using the same 莱雅公司 2023-06-27 CN disclosed
EP-2773633-B1 HETEROCYCLIC COMPOUNDS, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF BOEHRINGER INGELHEIM INT (DE) 2017-08-02 EP disclosed
US-8759349-B2 Heterocyclic compounds, medicaments containing said compounds, use thereof and processes for the preparation thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-06-24 US disclosed
WO-2013064450-A1 HETEROCYCLIC COMPOUNDS, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-05-10 WO disclosed
US-20130109697-A1 HETEROCYCLIC COMPOUNDS, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-05-02 US disclosed
EP-2322173-A1 Cationic bacteriochlorophyll derivatives and uses thereof YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 2011-05-18 EP disclosed
US-20100022483-A1 Substituted Tetracycline Compounds PARATEK PHARMACEUTICALS, INC. (US) 2010-01-28 US disclosed
WO-2008044099-A1 CHARGE TRANSFER COMPLEXES IN THE TREATMENT OF INFLAMMATORY BOWEL DISEASES GHISALBERTI CARLO (BR) 2008-04-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109697-A1 HETEROCYCLIC COMPOUNDS, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF SCNN1B, SCNN1A, TRPM5 KDM4E 4403/4885MAPK1 1581/4885HIF1A 1256/4885
US-20100022483-A1 Substituted Tetracycline Compounds TET1, TET3, TLR5 KDM4E 1796/4885MAPK1 4471/4885HIF1A 2040/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.