SCHEMBL183930

SCHEMBL183930

NC(=O)c1cc(F)ccc1N

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.70
IKBKB O14920 5/20 0.53
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
ALDH1A1 P00352 1/20 0.48
FADS1 O60427 1/20 0.47
PARP1 P09874 2/20 0.45
CHUK O15111 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
DGAT1 O75907 1/20 0.42
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 2/20 0.42
GFER P55789 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MEN1 O00255 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31230207 1.00 KEAP1 (0.70) KEAP1IKBKBCES2CES1ALDH1A1
Hydrochloric Acid SCHEMBL4362930 0.98 KEAP1 (0.68) KEAP1IKBKBCES2CES1ALDH1A1
Anthranilamide SCHEMBL4012579 0.91 KEAP1 (0.59) KEAP1IKBKBCES2CES1ALDH1A1
SCHEMBL5308529 0.84 IKBKB (0.71) KEAP1IKBKBCHUKCYP1A2CYP3A4
SCHEMBL135091 0.83 KEAP1 (1.00) KEAP1CES2CES1ALDH1A1FADS1
SCHEMBL29364785 0.83 KEAP1 (1.00) KEAP1CES2CES1ALDH1A1FADS1
SCHEMBL148542 0.83 KEAP1 (0.53) KEAP1IKBKBCES2CES1ALDH1A1
SCHEMBL29463969 0.82 CES2 (0.52) KEAP1IKBKBCES2CES1ALDH1A1
SCHEMBL12070396 0.82 KEAP1 (0.63) KEAP1IKBKBCES2CES1ALDH1A1
SCHEMBL9000281 0.81 KEAP1 (0.96) KEAP1CES2CES1ALDH1A1FADS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 212 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122010957-A Preparation method of fullerene pyrrolidine quinazolinone 湖北大学 2026-05-12 CN claimed
CN-120079371-A Oxygen vacancy-containing tungsten trioxide catalyst and preparation method and application thereof 南京理工大学 2025-06-03 CN claimed
EP-4746972-A1 DEUTERATED PARP1 INHIBITOR COMPOUNDS Duke Street Bio Limited (GB) 2026-05-27 EP disclosed
US-20260137684-A1 ROCK2 Inhibitors And Uses Thereof RESTOR PHARMACEUTICALS (US) 2026-05-21 US disclosed
WO-2026104681-A1 NEW SULFONAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2026-05-21 WO disclosed
CN-122055367-A 5-Oxo-4, 5-dihydroimidazo [1,5-a ] quinazoline compounds as PI3K [ alpha ] inhibitors 皮卡维森治疗学股份有限公司 2026-05-15 CN disclosed
CN-122010957-A Preparation method of fullerene pyrrolidine quinazolinone 湖北大学 2026-05-12 CN disclosed
EP-4127157-B1 MODIFIED DIPEPTIDE CLEAVASES, USES THEREOF AND RELATED KITS ENCODIA INC (US) 2026-02-11 EP disclosed
EP-4674841-A2 PHARMACEUTICAL COMPOUND Duke Street Bio Limited (GB) 2026-01-07 EP disclosed
CN-120079371-A Oxygen vacancy-containing tungsten trioxide catalyst and preparation method and application thereof 南京理工大学 2025-06-03 CN disclosed
WO-2025085474-A1 5-OXO-4,5-DIHYDROIMIDAZO[1,5-A]QUINAZOLINE COMPOUNDS AS PI3K[ALPHA] INHIBITORS SYNNOVATION THERAPEUTICS, INC. (US) 2025-04-24 WO disclosed
US-20050176955-A1 N-(substituted benzyl)-8-hydroxy-1,6-naphthyridine-7-carboxamides useful as hiv integrase inhibitors MERCK SHARP & DOHME CORP. 2005-08-11 US disclosed
WO-2005014585-A1 HALOGENATED QUINAZOLINYL NITROFURANS AS ANTIBACTERIAL AGENTS ULYSSES PHARMACEUTICAL PRODUCTS INC. (CA) 2005-02-17 WO disclosed
EP-1496836-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2004080402-A2 POTASSIUM SALT OF AN HIV INTEGRASE INHIBITOR MERCK & CO. INC. (US) 2004-09-23 WO disclosed
CN-1143855-C I (ortho)-anthranilamide derivatives as anti-coagulants ���ֹɷݹ�˾ 2004-03-31 CN disclosed
WO-2003077850-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed
WO-2003077857-A2 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2003-09-25 WO disclosed
US-6479499-B1 INHIBITORS OF TUBULIN POLYMERIZATION NATIONAL SCIENCE COUNCIL (TW) 2002-11-12 US disclosed
CN-1282329-A I (ortho)-anthranilamide derivatives as anti-coagulants SCHERING AG (DE) 2001-01-31 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176955-A1 N-(substituted benzyl)-8-hydroxy-1,6-naphthyridine-7-carboxamides useful as hiv integrase inhibitors CDK8, PNP, HINT1 KEAP1 3955/4885IKBKB 176/4885CES2 526/4885
US-20260137684-A1 ROCK2 Inhibitors And Uses Thereof ROCK2, ROCK1, RHOA KEAP1 1607/4885IKBKB 1656/4885CES2 976/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.