SCHEMBL18409178

SCHEMBL18409178

CCc1cc(C2=CCN(S(C)(=O)=O)CC2)ccc1N

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 4/20 0.52
MMP3 P08254 4/20 0.52
CCNT1 O60563 9/20 0.45
CDK9 P50750 9/20 0.45
TDO2 P48775 1/20 0.42
LMNA P02545 1/20 0.41
THRB P10828 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
ENPP2 Q13822 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14320646 0.81 TDO2 (0.49) MMP2MMP3CCNT1CDK9TDO2
SCHEMBL18409125 0.78 CCNT1 (0.45) CCNT1CDK9TDO2GPR119
SCHEMBL11956930 0.77 LMNA (0.62) MMP2MMP3CCNT1CDK9TDO2
SCHEMBL15174850 0.77 QDPR (0.49) MMP2MMP3L3MBTL1ALDH1A1
SCHEMBL979744 0.75 THRB (0.49) MMP2MMP3CCNT1CDK9TDO2
SCHEMBL979793 0.75 QDPR (0.58) MMP2MMP3CCNT1CDK9TDO2
SCHEMBL15615751 0.75 CCNT1 (0.49) CCNT1CDK9TDO2LMNATHRB
SCHEMBL24721518 0.74 MMP2 (0.56) MMP2MMP3CCNT1CDK9TDO2
SCHEMBL6437476 0.74 MMP2 (0.49) MMP2MMP3CCNT1CDK9TDO2
SCHEMBL979623 0.73 CCNT1 (0.49) MMP2MMP3CCNT1CDK9TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017012647-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2017-01-26 WO disclosed