SCHEMBL979623

SCHEMBL979623

CS(=O)(=O)N1CC=C(c2ccc(O)c(F)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 10/20 0.49
CDK9 P50750 10/20 0.49
MMP2 P08253 1/20 0.48
MMP3 P08254 1/20 0.48
LMNA P02545 1/20 0.48
THRB P10828 1/20 0.48
QDPR P09417 4/20 0.48
KDM4E B2RXH2 1/20 0.43
TDO2 P48775 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067599 0.85 CCNT1 (0.47) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL978744 0.82 CCNT1 (0.63) CCNT1CDK9LMNATHRB
SCHEMBL979793 0.82 QDPR (0.58) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL979744 0.79 THRB (0.49) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL11956930 0.78 LMNA (0.62) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL14320646 0.76 TDO2 (0.49) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL15615751 0.76 CCNT1 (0.49) CCNT1CDK9LMNATHRBKDM4E
SCHEMBL24721518 0.75 MMP2 (0.56) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL6437476 0.75 MMP2 (0.49) CCNT1CDK9MMP2MMP3LMNA
SCHEMBL1103889 0.73 CCNT1 (0.59) CCNT1CDK9MMP2MMP3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8207344-B2 GPR119 agonists ELI LILLY AND COMPANY (US) 2012-06-26 US disclosed
EP-2454251-A1 GPR119 AGONISTS Eli Lilly and Company (US) 2012-05-23 EP disclosed
CN-102432598-A Tricyclic compound, preparation method thereof and pharmaceutical application thereof JIANGSU HENGRUI MEDICINE CO 2012-05-02 CN disclosed
WO-2011008663-A1 GPR119 AGONISTS ELI LILLY AND COMPANY (US) 2011-01-20 WO disclosed
US-20110015199-A1 GPR119 Agonists ELI LILLY AND COMPANY (US) 2011-01-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110015199-A1 GPR119 Agonists GPR119, GLP1R, GCGR CCNT1 4475/4885CDK9 2128/4885MMP2 3487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.