SCHEMBL184592

SCHEMBL184592

O=C(O)C(Oc1ccc(Cl)c(Cl)c1)c1ccc(S(=O)(=O)C2CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GCK P35557 10/20 0.51
PPARG P37231 5/20 0.40
PPARA Q07869 2/20 0.40
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
F10 P00742 1/20 0.37
PLG P00747 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184497 0.90 GCK (0.51) GCKPPARGPPARA
SCHEMBL184498 0.88 GCK (0.63) GCKPPARGPPARA
SCHEMBL184640 0.83 GCK (0.50) GCKPPARG
SCHEMBL185010 0.83 GCK (0.48) GCKPPARGPPARA
SCHEMBL184731 0.82 GCK (0.50) GCK
SCHEMBL184906 0.82 MMP13 (0.51) GCKMMP2MMP9F10PRSS1
SCHEMBL197390 0.82 GCK (0.50) GCK
SCHEMBL185529 0.80 GCK (0.48) GCKPPARGPPARA
SCHEMBL184678 0.80 GCK (0.43) GCKPPARG
SCHEMBL184337 0.80 GCK (0.49) GCKPPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402327-B1 Acetamide compounds as glucokinase activators, their process and medicinal applications IMPETIS BIOSCIENCES LTD (IN) 2018-03-07 EP disclosed
EP-2402327-A1 Acetamide compounds as glucokinase activators, their process and medicinal applications Advinus Therapeutics Private Limited (IN) 2012-01-04 EP disclosed