SCHEMBL184498

SCHEMBL184498

O=C(O)C(Oc1ccc(Cl)cc1)c1ccc(S(=O)(=O)C2CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GCK P35557 9/20 0.63
PPARG P37231 7/20 0.46
PPARA Q07869 4/20 0.44
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
CASP3 P42574 1/20 0.39
KMT2A Q03164 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
ELOVL6 Q9H5J4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184640 0.88 GCK (0.50) GCKPPARGELOVL6
SCHEMBL184592 0.88 GCK (0.51) GCKPPARGPPARA
SCHEMBL184731 0.87 GCK (0.50) GCKKMT2AKEAP1NFE2L2ELOVL6
SCHEMBL184906 0.87 MMP13 (0.51) GCKKEAP1NFE2L2ELOVL6
SCHEMBL197390 0.87 GCK (0.50) GCKKEAP1NFE2L2
SCHEMBL184497 0.87 GCK (0.51) GCKPPARGPPARA
SCHEMBL185010 0.85 GCK (0.48) GCKPPARGPPARA
SCHEMBL185529 0.84 GCK (0.48) GCKPPARGPPARAKEAP1NFE2L2
SCHEMBL184976 0.84 GCK (0.48) GCKPPARGMEN1KMT2AKEAP1
SCHEMBL11748683 0.82 PPARG (0.51) GCKPPARGPPARAMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402327-B1 Acetamide compounds as glucokinase activators, their process and medicinal applications IMPETIS BIOSCIENCES LTD (IN) 2018-03-07 EP disclosed
EP-2402327-A1 Acetamide compounds as glucokinase activators, their process and medicinal applications Advinus Therapeutics Private Limited (IN) 2012-01-04 EP disclosed