SCHEMBL197390

SCHEMBL197390

O=C(O)C(Oc1ccc(F)cc1)c1ccc(S(=O)(=O)C2CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GCK P35557 15/20 0.50
HTR2A P28223 3/20 0.41
HTR2C P28335 2/20 0.41
KCNH2 Q12809 2/20 0.41
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184640 0.88 GCK (0.50) GCK
SCHEMBL185010 0.88 GCK (0.48) GCK
SCHEMBL184906 0.87 MMP13 (0.51) GCKKEAP1NFE2L2
SCHEMBL184498 0.87 GCK (0.63) GCKKEAP1NFE2L2
SCHEMBL184731 0.87 GCK (0.50) GCKKEAP1NFE2L2
SCHEMBL184976 0.86 GCK (0.48) GCKKEAP1NFE2L2
SCHEMBL185529 0.86 GCK (0.48) GCKKEAP1NFE2L2
SCHEMBL184337 0.86 GCK (0.49) GCK
SCHEMBL184497 0.84 GCK (0.51) GCK
SCHEMBL185100 0.83 GCK (0.66) GCKHTR2AHTR2CKCNH2KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402327-B1 Acetamide compounds as glucokinase activators, their process and medicinal applications IMPETIS BIOSCIENCES LTD (IN) 2018-03-07 EP disclosed
EP-2402327-A1 Acetamide compounds as glucokinase activators, their process and medicinal applications Advinus Therapeutics Private Limited (IN) 2012-01-04 EP disclosed