SCHEMBL18508977

SCHEMBL18508977

C=CNCc1ccc(C(=C)Cl)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.35
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20194348 0.71 HSD17B1 (0.33)
SCHEMBL11831189 0.70 SLC22A12 (0.37) NR1H4ESR1ESR2
SCHEMBL20428093 0.69 AXL (0.33)
SCHEMBL23373028 0.69 ADH1B (0.42)
SCHEMBL21696535 0.68 SMN1; SMN2 (0.46) HPGD
SCHEMBL11601038 0.68 TDP1 (0.44)
SCHEMBL23482035 0.68 ALDH1A1 (0.33)
SCHEMBL15275916 0.65 CES2 (0.38)
SCHEMBL15434406 0.64 MEN1 (0.52) HPGD
SCHEMBL23585808 0.64 LMNA (0.47) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2168952-B1 MORPHOLINE DERIVATIVES AS RENIN INHIBITORS MITSUBISHI TANABE PHARMA CORP (JP) 2017-02-15 EP disclosed