Bromide

Bromide

SCHEMBL1852155

Cc1c(Cc2cccc(C(F)(F)F)c2)oc2cccc(O)c12.[B+3].[Br-].[Br-].[Br-]

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.54
HTR2B P41595 3/20 0.50
GPR52 Q9Y2T5 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
AR P10275 1/20 0.40
MAOB P27338 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
MAPT P10636 3/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ACP3 P15309 1/20 0.38
CCR4 P51679 1/20 0.38
SLC26A3 P40879 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1848567 0.97 ALOX5 (0.56) ALOX5HTR2BGPR52MTNR1AMTNR1B
SCHEMBL1852157 0.93 ALOX5 (0.52) ALOX5HTR2BGPR52MTNR1AMTNR1B
SCHEMBL1849327 0.81 MTNR1A (0.46) ALOX5HTR2BGPR52MTNR1AMTNR1B
SCHEMBL3198348 0.78 MAOB (0.40) ALOX5HTR2BGPR52MTNR1AMTNR1B
SCHEMBL1848465 0.75 MAOB (0.38) ALOX5HTR2BGPR52MTNR1AMTNR1B
SCHEMBL1852178 0.75 GPR52 (0.56) GPR52MTNR1AMTNR1B
SCHEMBL1857128 0.71 HTR2B (0.47) HTR2BMAPTKMT2ATDP1ACP3
SCHEMBL9740770 0.70 ALOX5 (1.00) ALOX5HTR2BHTR2CMAPTNPC1
SCHEMBL1855422 0.69 GPR52 (0.53) HTR2BGPR52MTNR1AMTNR1BMAOB
SCHEMBL10744144 0.69 ALOX5 (0.57) ALOX5HTR2BARHTR2CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323978-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-05-25 EP disclosed
WO-2010018874-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed