SCHEMBL18569860

SCHEMBL18569860

C#CCn1cc(P)ccc1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
ADORA2B P29275 1/20 0.34
POLB P06746 2/20 0.31
HSP90AA1 P07900 1/20 0.31
PADI4 Q9UM07 1/20 0.30
CA12 O43570 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16220653 0.77 ALDH1A1 (0.53) MEN1KMT2AALDH1A1MAPTMAOA
SCHEMBL16194600 0.74 MEN1 (0.38) MEN1KMT2AALDH1A1MAPTMAOA
SCHEMBL27397709 0.65 ALDH1A1 (0.43) MEN1KMT2AALDH1A1MAPTMAOA
SCHEMBL26926255 0.60 HSD17B13 (0.50) ADORA2B
SCHEMBL379033 0.58 MAOA (0.47) ALDH1A1MAPTMAOAMAOBHSP90AA1
SCHEMBL22144561 0.58 PKM (0.47) ALDH1A1
SCHEMBL9521247 0.58 ADORA2B (0.34) MEN1KMT2AALDH1A1MAPTADORA2B
SCHEMBL9409708 0.56 ADORA2B (0.42) KMT2AMAOAMAOBADORA2B
SCHEMBL9409690 0.56
SCHEMBL9519935 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991981-B1 DIAMINOPYRAZINE COMPOUNDS, MEDICAMENTS CONTAINING SAID COMPOUNDS, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF BOEHRINGER INGELHEIM INT (DE) 2017-03-01 EP disclosed