SCHEMBL18640786

SCHEMBL18640786

Nc1nccc2c1C(=O)CCC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.52
NOS2 P35228 3/20 0.52
NOS1 P29475 1/20 0.52
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
CYP2A6 P11509 1/20 0.37
BUB1 O43683 4/20 0.34
PRKCI P41743 1/20 0.33
KDM4E B2RXH2 1/20 0.32
FGFR1 P11362 2/20 0.32
CHEK1 O14757 1/20 0.32
DAPK3 O43293 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32
CSF1R P07333 1/20 0.32
RET P07949 1/20 0.32
FLT1 P17948 1/20 0.32
LTK P29376 1/20 0.32
GRK5 P34947 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23566387 0.89 NOS3 (0.46) NOS3NOS2NOS1FGFR1CHEK1
SCHEMBL8295015 0.79 MAOA (0.38) NOS3NOS2NOS1MAOAMAOB
SCHEMBL19152890 0.78 BRD4 (0.37) NOS3NOS2NOS1MAOAMAOB
SCHEMBL27999392 0.78 MAOA (0.37) NOS3NOS2NOS1MAOAMAOB
SCHEMBL20478847 0.74 ALDH1A1 (0.36) NOS3NOS2NOS1MAOAMAOB
SCHEMBL18237671 0.74 MAOA (0.34) NOS3NOS2NOS1MAOAMAOB
SCHEMBL18640762 0.73 CHEK1 (0.49) NOS3NOS2NOS1FGFR1CHEK1
SCHEMBL16658453 0.72 NOS2 (0.92) NOS3NOS2NOS1LIMK1SIGMAR1
SCHEMBL23566352 0.71 NOS3 (0.41) NOS3NOS2NOS1MAOAMAOB
SCHEMBL23566363 0.71 NOS3 (0.41) NOS3NOS2NOS1FGFR1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3362436-B1 PROCESS FOR THE CATALYTIC DIRECTED CLEAVAGE OF AMIDE-CONTAINING COMPOUNDS UNIV ANTWERPEN (BE) 2021-06-30 EP claimed
EP-3362436-B1 PROCESS FOR THE CATALYTIC DIRECTED CLEAVAGE OF AMIDE-CONTAINING COMPOUNDS UNIV ANTWERPEN (BE) 2021-06-30 EP disclosed
EP-3362436-A1 PROCESS FOR THE CATALYTIC DIRECTED CLEAVAGE OF AMIDE-CONTAINING COMPOUNDS Universiteit Antwerpen (BE) 2018-08-22 EP disclosed
WO-2017046133-A1 PROCESS FOR THE CATALYTIC DIRECTED CLEAVAGE OF AMIDE-CONTAINING COMPOUNDS UNIVERSITEIT ANTWERPEN (BE) 2017-03-23 WO disclosed