SCHEMBL1867735

SCHEMBL1867735

CN1CCC(C(=O)NCc2cc[c]cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.53
ALDH1A1 P00352 5/20 0.50
USP2 O75604 1/20 0.50
HPGD P15428 1/20 0.50
TDP1 Q9NUW8 2/20 0.48
TSHR P16473 2/20 0.47
CYP3A4 P08684 1/20 0.47
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HTR1A P08908 1/20 0.47
HTR1B P28222 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23360779 0.86 ALDH1A1 (0.60) NPSR1ALDH1A1USP2HPGDSMN1; SMN2
SCHEMBL13746186 0.85 NPSR1 (0.72) NPSR1ALDH1A1USP2HPGDTDP1
SCHEMBL8372164 0.84 MEN1 (0.61) NPSR1ALDH1A1USP2HPGDTSHR
SCHEMBL12993901 0.84 ALDH1A1 (0.67) ALDH1A1USP2TDP1TSHRCYP3A4
SCHEMBL3321589 0.84 NPSR1 (0.52) NPSR1ALDH1A1USP2HPGDTSHR
SCHEMBL27734242 0.83 ALDH1A1 (0.66) NPSR1ALDH1A1USP2HPGDCYP3A4
SCHEMBL13745563 0.83 ALDH1A1 (0.67) NPSR1ALDH1A1TSHRCYP3A4LMNA
SCHEMBL13745754 0.83 ALDH1A1 (0.62) ALDH1A1
SCHEMBL13061265 0.83 ALDH1A1 (0.62) NPSR1ALDH1A1TSHRSMN1; SMN2
SCHEMBL13745506 0.81 ALDH1A1 (0.70) ALDH1A1TDP1TSHRLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008079988-A9 QUINAZOLINES FOR PDK1 INHIBITION NOVARTIS AG (CH) 2011-05-12 WO disclosed
US-20100216767-A1 QUINAZOLINES FOR PDK1 INHIBITION AIKAWA MINA 2010-08-26 US disclosed
US-20100121052-A1 Novel compounds for treating proliferative diseases JAIN RAMA 2010-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100216767-A1 QUINAZOLINES FOR PDK1 INHIBITION PDK1, PDK2, PDK3 NPSR1 4272/4885ALDH1A1 2630/4885USP2 2578/4885
US-20100121052-A1 Novel compounds for treating proliferative diseases PDK1, PDK2, PDK3 NPSR1 4212/4885ALDH1A1 2281/4885USP2 2868/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.