SCHEMBL18840973

SCHEMBL18840973

CCOC(=O)c1cnn(CC(O)c2ccccc2)c1NC(=O)Nc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
LMNA P02545 1/20 0.47
HTT P42858 3/20 0.45
RAB9A P51151 2/20 0.45
KDM4E B2RXH2 3/20 0.44
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PDE4B Q07343 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
KDR P35968 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
CASR P41180 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18840958 0.89 ALDH1A1 (0.48) ALDH1A1LMNAHTTRAB9AKDM4E
SCHEMBL18840970 0.87 MAPT (0.48) ALDH1A1LMNAHTTRAB9AKDM4E
SCHEMBL4075658 0.86 ALDH1A1 (0.47) ALDH1A1LMNAKDM4EMAPTADORA1
SCHEMBL8693084 0.83 ALDH1A1 (0.54) ALDH1A1LMNAHTTRAB9AKDM4E
SCHEMBL3868209 0.82 ALDH1A1 (0.52) ALDH1A1LMNAHTTRAB9AKDM4E
SCHEMBL8696943 0.80 ALDH1A1 (0.54) ALDH1A1LMNAHTTRAB9AKDM4E
SCHEMBL4075047 0.80 MAPT (0.53) ALDH1A1LMNARAB9AKDM4EMAPT
SCHEMBL4067165 0.80 MAPT (0.53) ALDH1A1LMNARAB9AKDM4EMAPT
SCHEMBL4070954 0.79 HPGD (0.60) ALDH1A1LMNAHTTRAB9AKDM4E
SCHEMBL31065210 0.79 PAX8 (0.54) LMNAHTTRAB9AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10401365-B2 Inhibition of chemokine CCL7 or receptor CCR3 of same for the treatment and diagnosis of prostate cancer UNIVERSITE PAUL SABATIER (TOULOUSE III) (FR) 2019-09-03 US disclosed
US-20170131282-A1 Inhibition of Chemokine CCL7 or Receptor CCR3 of Same for the Treatment and Diagnosis of Prostate Cancer INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2017-05-11 US disclosed
US-20170131282-A1 Inhibition of Chemokine CCL7 or Receptor CCR3 of Same for the Treatment and Diagnosis of Prostate Cancer INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2017-05-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170131282-A1 Inhibition of Chemokine CCL7 or Receptor CCR3 of Same for the Treatment and Diagnosis of Prostate Cancer CCR3, CCR5, CCR1 ALDH1A1 1318/4885LMNA 4732/4885HTT 4688/4885
US-10401365-B2 Inhibition of chemokine CCL7 or receptor CCR3 of same for the treatment and diagnosis of prostate cancer CCR3, CCR5, CCR1 ALDH1A1 1281/4885LMNA 4728/4885HTT 4699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.