SCHEMBL18900166

SCHEMBL18900166

CCC(=O)Nc1ccnc(C)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 4/20 0.50
ADORA3 P0DMS8 9/20 0.46
ADORA1 P30542 6/20 0.46
ADORA2A P29274 5/20 0.46
ADORA2B P29275 4/20 0.46
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
TYK2 P29597 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
POLB P06746 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GRM5 P41594 1/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RIPK1 Q13546 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1428795 0.85 SORT1 (0.52) SORT1GRM5SMN1; SMN2RIPK1ALDH1A1
SCHEMBL4551723 0.83 CA1 (0.47) ADORA3ADORA1ADORA2AADORA2BJAK2
SCHEMBL20068960 0.80 SORT1 (0.54) SORT1ADORA3ADORA2AADORA2BPOLB
SCHEMBL19150881 0.79 ADORA3 (0.46) ADORA3ADORA1ADORA2AADORA2BJAK2
SCHEMBL19151254 0.78 CTSK (0.44) ADORA3ADORA1ADORA2AADORA2BJAK2
SCHEMBL14667358 0.76 CYP1A2 (0.56) SORT1ADORA1POLBGRM5RIPK1
SCHEMBL8240613 0.76 RAB9A (0.59) NPC1RAB9APOLBTP53SMN1; SMN2
SCHEMBL13922914 0.76 RAB9A (0.59) NPC1RAB9APOLBTP53SMN1; SMN2
SCHEMBL4551457 0.76 SMN1; SMN2 (0.65) ADORA3ADORA1ADORA2AADORA2BNPC1
SCHEMBL19176885 0.75 ATM (0.48) SORT1POLBTDP1GRM5RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651899-B1 SUBSTITUTED 6,6-FUSED NITROGENOUS HETEROCYCLIC COMPOUNDS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2017-05-31 EP disclosed