SCHEMBL1894516

SCHEMBL1894516

O=C(Oc1c(F)c(F)c(F)c(F)c1F)c1ncccc1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 5/20 0.43
EGLN2 Q96KS0 1/20 0.42
FTO Q9C0B1 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 4/20 0.37
SPR P35270 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
BLM P54132 1/20 0.36
AGER Q15109 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
BRD4 O60885 1/20 0.35
NAPRT Q6XQN6 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31645626 0.83 ALDH1A1 (0.42) L3MBTL1KDM4EALDH1A1CYP3A4MAPT
SCHEMBL108876 0.78 L3MBTL1 (0.62) TLR7EGLN2FTOL3MBTL1KDM4E
SCHEMBL28048185 0.78 TLR7 (0.48) TLR7EGLN2FTOL3MBTL1KDM4E
SCHEMBL2304193 0.76 LMNA (0.35) TLR7L3MBTL1KDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL6569637 0.76 L3MBTL1 (0.60) TLR7EGLN2FTOL3MBTL1KDM4E
SCHEMBL31646056 0.76 FEN1 (0.50) L3MBTL1KDM4EALDH1A1
SCHEMBL27832422 0.75 EGLN2 (0.49) TLR7EGLN2FTOL3MBTL1KDM4E
SCHEMBL7833009 0.75 L3MBTL1 (0.51) TLR7EGLN2FTOL3MBTL1KDM4E
SCHEMBL31645520 0.74 GRM5 (0.43) KDM4EALDH1A1CYP3A4MAPTALOX15
SCHEMBL1829785 0.74 KDM4E (0.47) TLR7EGLN2FTOL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025137640-A1 AZASPIRO WRN INHIBITORS GILEAD SCIENCES, INC. (US) 2025-06-26 WO disclosed
EP-4347596-A1 TRIAZOLO-PYRIMIDINE ANALOGUES FOR TREATING DISEASES CONNECTED TO THE INHIBITON OF WERNER SYNDROME RECQ HELICASE (WRN) Novartis AG (CH) 2024-04-10 EP disclosed
US-20230046859-A1 Bicyclic Compounds and their Uses NOVARTIS PHARMA AG (CH) 2023-02-16 US disclosed
WO-2022249060-A1 TRIAZOLO-PYRIMIDINE ANALOGUES FOR TREATING DISEASES CONNECTED TO THE INHIBITON OF WERNER SYNDROME RECQ HELICASE (WRN) NOVARTIS AG (CH) 2022-12-01 WO disclosed
EP-2718298-A1 SUBSTITUTED PYRIDINES HAVING HERBICIDAL ACTIVITY BASF SE (DE) 2014-04-16 EP disclosed
US-8338337-B2 Substituted pyridines having a herbicidal effect BASF SE (DE) 2012-12-25 US disclosed
WO-2012168397-A1 SUBSTITUTED PYRIDINES HAVING HERBICIDAL ACTIVITY BASF SE (DE) 2012-12-13 WO disclosed
WO-2012168397-A1 SUBSTITUTED PYRIDINES HAVING HERBICIDAL ACTIVITY BASF SE (DE) 2012-12-13 WO disclosed
US-20110224078-A1 Substituted Pyridines Having a Herbicidal Effect BASF SE (DE) 2011-09-15 US disclosed
US-20110201501-A1 Substituted Pyridines Having a Herbicidal Effect BASF SE (DE) 2011-08-18 US disclosed
WO-2011057942-A1 INSECTICIDAL METHODS USING PYRIDINE COMPOUNDS BASF SE (DE) 2011-05-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110201501-A1 Substituted Pyridines Having a Herbicidal Effect DDT, PNPO, HPD TLR7 3745/4885EGLN2 570/4885FTO 424/4885
US-20230046859-A1 Bicyclic Compounds and their Uses H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, C1R, F12 TLR7 196/4885EGLN2 2974/4885FTO 3943/4885
US-20110224078-A1 Substituted Pyridines Having a Herbicidal Effect DDT, PNPO, HPD TLR7 3745/4885EGLN2 570/4885FTO 424/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.